Compile Data Set for Download or QSAR
maximum 50k data
Report error Found 179 Enz. Inhib. hit(s) with all data for entry = 50035685
LigandPNGBDBM50367516(CHEMBL1907724)
Affinity DataIC50:  100nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM82388(CCK antagonist synthetic 11)
Affinity DataIC50:  270nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367541(CHEMBL1907742)
Affinity DataIC50:  300nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367530(CHEMBL1907731)
Affinity DataIC50:  300nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM82392(CCK antagonist synthetic 13)
Affinity DataIC50:  300nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367523(CHEMBL1907729)
Affinity DataIC50:  360nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM82393(CCK antagonist synthetic 9)
Affinity DataIC50:  500nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367518(CHEMBL1907720)
Affinity DataIC50:  700nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM82391(CCK antagonist synthetic 8)
Affinity DataIC50:  1.20E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50023140(6-(2-Fluoro-phenyl)-4-(1H-indol-3-ylmethyl)-1-meth...)
Affinity DataIC50:  1.20E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019812(3-(6-Fluoro-1H-indol-3-ylmethyl)-5-(2-fluoro-pheny...)
Affinity DataIC50:  1.30E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019777(7-(9-Hydroxy-2-isobutyl-3-oxo-2,3,9,9a-tetrahydro-...)
Affinity DataIC50:  1.40E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019804(3-(5-Fluoro-1H-indol-3-ylmethyl)-5-(2-fluoro-pheny...)
Affinity DataIC50:  1.40E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019785((R)7-Chloro-3-(1H-indol-3-ylmethyl)-5-phenyl-1,3-d...)
Affinity DataIC50:  1.40E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367544(CHEMBL1907719)
Affinity DataIC50:  1.40E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367526(CHEMBL1907725)
Affinity DataIC50:  2.10E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367533(CHEMBL1907737)
Affinity DataIC50:  2.20E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50226859(CHEMBL283946)
Affinity DataIC50:  2.90E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50421831(CHEMBL2092748)
Affinity DataIC50:  3.20E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019202(7-Chloro-3-(1H-indol-3-ylmethyl)-5-phenyl-1,3-dihy...)
Affinity DataIC50:  3.40E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367529(CHEMBL1907716)
Affinity DataIC50:  3.60E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367528(CHEMBL1907738)
Affinity DataIC50:  4.00E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367537(CHEMBL1907744)
Affinity DataIC50:  4.50E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019802((R alpha/beta) {3-Methyl-1-[3-(2-oxo-5-phenyl-2,3-...)
Affinity DataIC50:  4.70E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367547(CHEMBL1907741)
Affinity DataIC50:  5.00E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM82392(CCK antagonist synthetic 13)
Affinity DataIC50:  5.00E+3nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367544(CHEMBL1907719)
Affinity DataIC50:  5.80E+3nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019821((R alpha/beta) 3-[1-(2-Amino-4-methyl-pentanoyl)-2...)
Affinity DataIC50:  6.60E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367539(CHEMBL1907730)
Affinity DataIC50:  8.30E+3nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM82388(CCK antagonist synthetic 11)
Affinity DataIC50:  1.00E+4nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to guinea pig brain(cortex) cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367526(CHEMBL1907725)
Affinity DataIC50: >1.00E+4nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019803((R alpha) 1-Methyl-3-(1-methyl-2,3-dihydro-1H-indo...)
Affinity DataIC50:  1.00E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50421827(CHEMBL2092746)
Affinity DataIC50:  1.00E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50367530(CHEMBL1907731)
Affinity DataIC50:  1.00E+4nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to guinea pig brain(cortex) cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367522(CHEMBL1907930)
Affinity DataIC50:  1.06E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50367544(CHEMBL1907719)
Affinity DataIC50:  1.10E+4nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to guinea pig brain(cortex) cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367532(CHEMBL1907721)
Affinity DataIC50:  1.10E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50421825(CHEMBL2092991)
Affinity DataIC50:  1.10E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50421826(CHEMBL2092988)
Affinity DataIC50:  1.10E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367521(CHEMBL1907726)
Affinity DataIC50:  1.20E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50023140(6-(2-Fluoro-phenyl)-4-(1H-indol-3-ylmethyl)-1-meth...)
Affinity DataIC50:  1.20E+4nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50421828(CHEMBL2092990)
Affinity DataIC50:  1.30E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367534(CHEMBL1907734)
Affinity DataIC50:  1.30E+4nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM82388(CCK antagonist synthetic 11)
Affinity DataIC50:  1.30E+4nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50367518(CHEMBL1907720)
Affinity DataIC50:  1.30E+4nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019803((R alpha) 1-Methyl-3-(1-methyl-2,3-dihydro-1H-indo...)
Affinity DataIC50:  1.40E+4nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50019797(5-(2-Fluoro-phenyl)-3-thiophen-3-ylmethyl-1,3-dihy...)
Affinity DataIC50:  1.40E+4nMAssay Description:Half-maximal inhibition of binding of [125I]gastrin to guinea pig gastric glandsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50367524(CHEMBL1907735)
Affinity DataIC50:  1.60E+4nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to guinea pig brain(cortex) cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

LigandPNGBDBM50421830(CHEMBL2092749)
Affinity DataIC50:  1.70E+4nMAssay Description:Half-maximal inhibition of [125I]-CCK-33 binding to rat pancreas cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetCholecystokinin receptor type A(Guinea pig)
TBA

Curated by ChEMBL
LigandPNGBDBM50367523(CHEMBL1907729)
Affinity DataIC50:  1.70E+4nMAssay Description:Half-maximal inhibition of [125I]CCK-33 binding to guinea pig brain(cortex) cholecystokinin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

Displayed 1 to 50 (of 179 total ) | Next | Last >>
Jump to: