TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 0.870nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 0.910nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 7.30nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 9nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Ability to inhibit [3H]spiperone binding to 5-hydroxytryptamine 2 receptor determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Ability to inhibit [3H]spiperone binding to 5-hydroxytryptamine 2 receptor determined in ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 57nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 250nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 310nMAssay Description:Ability to inhibit [3H]spiperone binding to 5-hydroxytryptamine 2 receptor determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 480nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 700nMAssay Description:Ability to inhibit [3H]spiperone binding to 5-hydroxytryptamine 2 receptor determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 1.10E+3nMAssay Description:Ability to inhibit the [3H]spiperone binding to striatum Dopamine receptor D2 was determined in ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.10E+3nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 9.30E+3nMAssay Description:Ability to inhibit [3H]spiperone binding to 5-hydroxytryptamine 2 receptor determined in ratMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Duphar Research Laboratories
Curated by ChEMBL
Duphar Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Ability to inhibit [3H]WB-4101 binding to alpha-1 adrenergic receptor was determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 2.70E+4nMAssay Description:Ability to inhibit [3H]spiperone binding to 5-hydroxytryptamine 2 receptor determined in ratMore data for this Ligand-Target Pair
Affinity DataKi: 5.40E+4nMAssay Description:Ability to inhibit [3H]spiperone binding to 5-hydroxytryptamine 2 receptor determined in ratMore data for this Ligand-Target Pair