TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 0.110nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 1.90nMAssay Description:Inhibition of human TEC using poly[Glu:Tyr] as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition by filter binding methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 7nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 8nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 18nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 44nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 77nMAssay Description:Inhibition of His-tagged full length recombinant human LCK expressed in baculovirus expression system using TK-substrate-biotin after 40 mins by HTRF...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 106nMAssay Description:Inhibition of His-tagged full length recombinant human LCK expressed in baculovirus expression system using TK-substrate-biotin after 40 mins by HTRF...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 137nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 153nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 271nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Tec(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 306nMAssay Description:Inhibition of human TEC using poly[Glu:Tyr] as substrate preincubated for 20 mins followed by [gamma-33P]-ATP addition by filter binding methodMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 334nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 337nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 468nMAssay Description:Inhibition of His-tagged full length recombinant human LCK expressed in baculovirus expression system using TK-substrate-biotin after 40 mins by HTRF...More data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lyn(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of recombinant human LYN using TK-substrate-biotin after 40 mins by HTRF assayMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 526nMAssay Description:Inhibition of Fibrinogen binding to Fibrinogen receptorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 531nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 1.21E+3nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase BTK(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 1.38E+3nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 8.82E+3nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 9.22E+3nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 1.44E+4nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetCytoplasmic tyrosine-protein kinase BMX(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 1.83E+4nMAssay Description:Inhibition of His-tagged full length recombinant human BMX expressed in baculovirus expression system using TK-substrate-biotin after 40 mins by HTRF...More data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 2.05E+4nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: 2.71E+4nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of ADP-induced platelet aggregation in human platelet-rich plasmaMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair
TargetMitogen-activated protein kinase 14(Homo sapiens (Human))
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
National Institute Of Biological Sciences, Beijing
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:The compound was tested for the inhibition of fibrinogen receptorMore data for this Ligand-Target Pair