Compile Data Set for Download or QSAR
Report error Found 82 Enz. Inhib. hit(s) with all data for entry = 50000432
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250205(CHEMBL4067491)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250201(CHEMBL4070639)
Affinity DataEC50:  1.40nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250206(CHEMBL4060816)
Affinity DataEC50:  1.80nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250201(CHEMBL4070639)
Affinity DataEC50:  2nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250214(CHEMBL4100598)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250200(CHEMBL4064777)
Affinity DataEC50:  2.80nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  3.10nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250204(CHEMBL4060937)
Affinity DataEC50:  3.20nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250205(CHEMBL4067491)
Affinity DataEC50:  5.70nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250203(CHEMBL4083755)
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50017181(CHEMBL441738)
Affinity DataEC50:  6.80nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250207(CHEMBL4082585)
Affinity DataEC50:  7.60nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  8.60nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  9.20nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250206(CHEMBL4060816)
Affinity DataEC50:  9.20nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250204(CHEMBL4060937)
Affinity DataEC50:  9.60nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250213(CHEMBL4104927)
Affinity DataEC50:  11nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250209(CHEMBL4090425)
Affinity DataEC50:  13nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  17nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250214(CHEMBL4100598)
Affinity DataEC50:  18nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250201(CHEMBL4070639)
Affinity DataEC50:  19nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  24nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250200(CHEMBL4064777)
Affinity DataEC50:  29nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250205(CHEMBL4067491)
Affinity DataEC50:  31nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  34nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50027084(Melatonan)
Affinity DataEC50:  34nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50029747((4S)-4-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-[({[(2S...)
Affinity DataEC50:  35nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250213(CHEMBL4104927)
Affinity DataEC50:  43nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250207(CHEMBL4082585)
Affinity DataEC50:  64nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250203(CHEMBL4083755)
Affinity DataEC50:  89nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250205(CHEMBL4067491)
Affinity DataEC50:  110nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250199(CHEMBL4092477)
Affinity DataEC50:  112nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250206(CHEMBL4060816)
Affinity DataEC50:  123nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250209(CHEMBL4090425)
Affinity DataEC50:  124nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250201(CHEMBL4070639)
Affinity DataEC50:  137nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250204(CHEMBL4060937)
Affinity DataEC50:  160nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250214(CHEMBL4100598)
Affinity DataEC50:  162nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250212(CHEMBL4089119)
Affinity DataEC50:  185nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250182(CHEMBL4077331)
Affinity DataEC50:  258nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250213(CHEMBL4104927)
Affinity DataEC50:  291nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250206(CHEMBL4060816)
Affinity DataEC50:  299nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250210(CHEMBL4087072)
Affinity DataEC50:  318nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250200(CHEMBL4064777)
Affinity DataEC50:  375nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 3(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250200(CHEMBL4064777)
Affinity DataEC50:  633nMAssay Description:Agonist activity at EYFP-fused human MC3R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 5(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250214(CHEMBL4100598)
Affinity DataEC50:  635nMAssay Description:Agonist activity at EYFP-fused human MC5R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250208(CHEMBL4062443)
Affinity DataEC50:  678nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells after 16 to 20 hrs by CRE-driven reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
TargetMelanocortin receptor 4(Human)
University of Copenhagen

Curated by ChEMBL
LigandPNGBDBM50250182(CHEMBL4077331)
Affinity DataEC50:  685nMAssay Description:Agonist activity at EYFP-fused human MC4R expressed in HEK293 cells assessed as increase in cAMP accumulation after 30 mins by luminescent enzymatic ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/21/2019
Entry Details Article
PubMed
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