Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with all data for entry = 50001414
TargetHistone deacetylase 8(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50005711(CHEBI:46024 | GNF-Pf-1011 | TRICHOSTATIN | Trichos...)
Affinity DataKi:  45nMAssay Description:Inhibition of C-terminal His-tagged human recombinant full-length HDAC8 expressed in baculovirus expression system assessed as reduction in 7-amino-4...More data for this Ligand-Target Pair
TargetHistone deacetylase 8(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM19149(CHEMBL98 | N-hydroxy-N'-phenyloctanediamide | SAHA...)
Affinity DataKi:  480nMAssay Description:The compound was tested in vitro for binding activity against M1 muscarinic receptor in homogenates of the cerebral cortex of rat using [3H]pirenzepi...More data for this Ligand-Target Pair
TargetHistone deacetylase(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50278967(CHEMBL4162981)
Affinity DataIC50:  2.92E+5nMAssay Description:Antagonist activity for rat histamine H3 receptor was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed