TargetEstrogen receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 85nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 67nMAssay Description:Binding affinity to recombinant human GFP-fused ERalpha LBD (301 to 553 residues) expressed in Escherichia coli BL21(DE3) after 40 mins in presence o...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 213nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 297nMAssay Description:Binding affinity to recombinant human GFP-fused ERbeta LBD (259 to 498 residues) expressed in Escherichia coli BL21(DE3) after 40 mins in presence of...More data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 82nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: >2.00E+3nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 142nMAssay Description:Binding affinity to recombinant human GST-tagged VDR LBD (156 to 453 residues) expressed in Echerichia coli BL21 star (DE3) after 40 mins in presence...More data for this Ligand-Target Pair
TargetVitamin D3 receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 197nMAssay Description:Binding affinity to recombinant human GST-tagged VDR LBD (156 to 453 residues) expressed in Echerichia coli BL21 star (DE3) after 40 mins in presence...More data for this Ligand-Target Pair
TargetEstrogen receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 118nMAssay Description:Binding affinity to recombinant human GFP-fused ERalpha LBD (301 to 553 residues) expressed in Escherichia coli BL21(DE3) after 40 mins in presence o...More data for this Ligand-Target Pair
TargetEstrogen receptor beta(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 270nMAssay Description:Binding affinity to recombinant human GFP-fused ERbeta LBD (259 to 498 residues) expressed in Escherichia coli BL21(DE3) after 40 mins in presence of...More data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 248nMAssay Description:Binding affinity to recombinant human GST-tagged PGR LBD (678 to 933 residues) expressed in Escherichia coli BL21 star(DE3) after 40 mins in presence...More data for this Ligand-Target Pair
TargetProgesterone receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Shenzhen Graduate School Of Peking University
Curated by ChEMBL
Affinity DataKd: 178nMAssay Description:Binding affinity to recombinant human GST-tagged PGR LBD (678 to 933 residues) expressed in Escherichia coli BL21 star(DE3) after 40 mins in presence...More data for this Ligand-Target Pair