Compile Data Set for Download or QSAR
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Found 12 Enz. Inhib. hit(s) with all data for entry = 50000193
TargetEstrogen receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242218(CHEMBL4086339)
Affinity DataKd:  85nMAssay Description:Inhibition of HIV-1 protease in 10% fetal calf serum(FCS)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242219(CHEMBL4067602)
Affinity DataKd:  67nMAssay Description:Binding affinity to recombinant human GFP-fused ERalpha LBD (301 to 553 residues) expressed in Escherichia coli BL21(DE3) after 40 mins in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242220(CHEMBL4066573)
Affinity DataKd:  213nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242219(CHEMBL4067602)
Affinity DataKd:  297nMAssay Description:Binding affinity to recombinant human GFP-fused ERbeta LBD (259 to 498 residues) expressed in Escherichia coli BL21(DE3) after 40 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242220(CHEMBL4066573)
Affinity DataKd:  82nMAssay Description:Inhibition of HIV-1 protease in 5%DMSOMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242219(CHEMBL4067602)
Affinity DataKd: >2.00E+3nMAssay Description:Inhibition of the binding of [3H]C18-Platelet activating factor to human platelet membrane preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242220(CHEMBL4066573)
Affinity DataKd:  142nMAssay Description:Binding affinity to recombinant human GST-tagged VDR LBD (156 to 453 residues) expressed in Echerichia coli BL21 star (DE3) after 40 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242218(CHEMBL4086339)
Affinity DataKd:  197nMAssay Description:Binding affinity to recombinant human GST-tagged VDR LBD (156 to 453 residues) expressed in Echerichia coli BL21 star (DE3) after 40 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242220(CHEMBL4066573)
Affinity DataKd:  118nMAssay Description:Binding affinity to recombinant human GFP-fused ERalpha LBD (301 to 553 residues) expressed in Escherichia coli BL21(DE3) after 40 mins in presence o...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEstrogen receptor beta(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242218(CHEMBL4086339)
Affinity DataKd:  270nMAssay Description:Binding affinity to recombinant human GFP-fused ERbeta LBD (259 to 498 residues) expressed in Escherichia coli BL21(DE3) after 40 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242219(CHEMBL4067602)
Affinity DataKd:  248nMAssay Description:Binding affinity to recombinant human GST-tagged PGR LBD (678 to 933 residues) expressed in Escherichia coli BL21 star(DE3) after 40 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Shenzhen Graduate School Of Peking University

Curated by ChEMBL
LigandPNGBDBM50242218(CHEMBL4086339)
Affinity DataKd:  178nMAssay Description:Binding affinity to recombinant human GST-tagged PGR LBD (678 to 933 residues) expressed in Escherichia coli BL21 star(DE3) after 40 mins in presence...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed