Compile Data Set for Download or QSAR
maximum 50k data
Found 62 Enz. Inhib. hit(s) with all data for entry = 50000444
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250403(CHEMBL2386454)
Affinity DataEC50:  8.26E+3nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250423(CHEMBL4105577)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250405(CHEMBL4065144)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250406(CHEMBL4092815)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250407(CHEMBL4085061)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250408(CHEMBL4095263)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250409(CHEMBL4074812)
Affinity DataEC50:  7.42E+3nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250410(CHEMBL4089458)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250411(CHEMBL4061465)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250412(CHEMBL4091234)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250413(CHEMBL4078865)
Affinity DataEC50:  2.58E+3nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250414(CHEMBL4086723)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250415(CHEMBL4065290)
Affinity DataEC50:  2.74E+3nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250416(CHEMBL4063373)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250417(CHEMBL4101433)
Affinity DataEC50:  3.58E+3nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250418(CHEMBL4073017)
Affinity DataEC50:  3.75E+3nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250419(CHEMBL4064434)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250420(CHEMBL4085969)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250421(CHEMBL4097843)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250423(CHEMBL4105577)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250424(CHEMBL4087701)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250433(CHEMBL4095394)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250413(CHEMBL4078865)
Affinity DataEC50:  2.12E+3nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250434(CHEMBL4103142)
Affinity DataEC50:  920nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250415(CHEMBL4065290)
Affinity DataEC50:  3.27E+3nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250403(CHEMBL2386454)
Affinity DataEC50:  3.17E+3nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250435(CHEMBL4100545)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250405(CHEMBL4065144)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250406(CHEMBL4092815)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250407(CHEMBL4085061)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250408(CHEMBL4095263)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250409(CHEMBL4074812)
Affinity DataEC50:  2.83E+3nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250410(CHEMBL4089458)
Affinity DataEC50:  7.12E+3nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250411(CHEMBL4061465)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250412(CHEMBL4091234)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250416(CHEMBL4063373)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250436(CHEMBL4083446)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250418(CHEMBL4073017)
Affinity DataEC50:  2.51E+3nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250437(CHEMBL4093716)
Affinity DataEC50:  4.89E+3nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250420(CHEMBL4085969)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250421(CHEMBL4097843)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250438(CHEMBL4079815)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250424(CHEMBL4087701)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250439(CHEMBL4068003)
Affinity DataEC50:  820nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250433(CHEMBL4095394)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250435(CHEMBL4100545)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250445(CHEMBL4103009)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250446(CHEMBL4061301)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of California

Curated by ChEMBL
LigandPNGBDBM50250447(CHEMBL4077062)
Affinity DataEC50: >1.00E+4nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Mus musculus)
University Of California

Curated by ChEMBL
LigandPNGBDBM50250434(CHEMBL4103142)
Affinity DataEC50:  2.01E+3nMAssay Description:Agonist activity at mouse TLR4 expressed in HEK293 blue cells assessed as induction of NF-kappaB activation-mediated SEAP production after 20 to 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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