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Report error Found 98 Enz. Inhib. hit(s) with all data for entry = 50000451
TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250586(CHEMBL4093140)
Affinity DataIC50:  0.0100nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134946(CHEMBL2370964 | H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Ar...)
Affinity DataIC50:  0.300nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250586(CHEMBL4093140)
Affinity DataIC50:  0.400nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250591(CHEMBL4072387)
Affinity DataIC50:  0.400nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250589(CHEMBL4060000)
Affinity DataIC50:  0.420nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50268806(Ac-Tyr-Val-Nle-Gly-His-DPhe-Arg-Trp-Asp-Arg-Phe-Gl...)
Affinity DataIC50:  0.5nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250590(CHEMBL4081900)
Affinity DataIC50:  1.10nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250585(CHEMBL4104092)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50268806(Ac-Tyr-Val-Nle-Gly-His-DPhe-Arg-Trp-Asp-Arg-Phe-Gl...)
Affinity DataIC50:  1.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50268806(Ac-Tyr-Val-Nle-Gly-His-DPhe-Arg-Trp-Asp-Arg-Phe-Gl...)
Affinity DataIC50:  2nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250586(CHEMBL4093140)
Affinity DataIC50:  2.20nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50268806(Ac-Tyr-Val-Nle-Gly-His-DPhe-Arg-Trp-Asp-Arg-Phe-Gl...)
Affinity DataIC50:  2.40nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250586(CHEMBL4093140)
Affinity DataIC50:  3.30nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134946(CHEMBL2370964 | H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Ar...)
Affinity DataIC50:  3.5nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250587(CHEMBL4079302)
Affinity DataIC50:  4.10nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134946(CHEMBL2370964 | H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Ar...)
Affinity DataIC50:  5nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250591(CHEMBL4072387)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250587(CHEMBL4079302)
Affinity DataIC50:  5nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50134946(CHEMBL2370964 | H-Tyr-Val-Nle-Gly-His-D-Nal(2')-Ar...)
Affinity DataIC50:  6nMAssay Description:Agonist activity at human MC4R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250590(CHEMBL4081900)
Affinity DataIC50:  6.70nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250589(CHEMBL4060000)
Affinity DataIC50:  16nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250581(CHEMBL4068475)
Affinity DataIC50:  17nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250587(CHEMBL4079302)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250588(CHEMBL4103570)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250591(CHEMBL4072387)
Affinity DataIC50:  18nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250583(CHEMBL4089770)
Affinity DataIC50:  20nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250583(CHEMBL4089770)
Affinity DataIC50:  23nMAssay Description:Agonist activity at human MC5R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250580(CHEMBL4088516)
Affinity DataIC50:  24nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250591(CHEMBL4072387)
Affinity DataIC50:  30nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250582(CHEMBL4068654)
Affinity DataIC50:  36nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250585(CHEMBL4104092)
Affinity DataIC50:  40nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250584(CHEMBL4090684)
Affinity DataIC50:  42nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250585(CHEMBL4104092)
Affinity DataIC50:  45nMAssay Description:Agonist activity at human MC1R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation measured after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250583(CHEMBL4089770)
Affinity DataIC50:  56nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250584(CHEMBL4090684)
Affinity DataIC50:  68nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50026883(CHEMBL437050)
Affinity DataIC50:  71nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250587(CHEMBL4079302)
Affinity DataIC50:  82nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250589(CHEMBL4060000)
Affinity DataIC50:  117nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250582(CHEMBL4068654)
Affinity DataIC50:  118nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250581(CHEMBL4068475)
Affinity DataIC50:  137nMAssay Description:Agonist activity at human MC3R expressed in HEK293 cells assessed as induction of intracellular cAMP accumulation after 3 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250580(CHEMBL4088516)
Affinity DataIC50:  210nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250583(CHEMBL4089770)
Affinity DataIC50:  254nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250585(CHEMBL4104092)
Affinity DataIC50:  330nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250582(CHEMBL4068654)
Affinity DataIC50:  360nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 4(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50026883(CHEMBL437050)
Affinity DataIC50:  760nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250580(CHEMBL4088516)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocyte-stimulating hormone receptor(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50026883(CHEMBL437050)
Affinity DataIC50:  1.00E+3nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC1R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250590(CHEMBL4081900)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 5(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250584(CHEMBL4090684)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC5R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetMelanocortin receptor 3(Human)
The University of Arizona

Curated by ChEMBL
LigandPNGBDBM50250584(CHEMBL4090684)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC3R expressed in HEK293 cells after 40 mins by gamma counting methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

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