Found 70 Enz. Inhib. hit(s) with all data for entry = 50001136 
Affinity DataEC50: 3.20nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 3.60nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 17nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 4.40nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 1.40nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 12nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 6nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 3.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 4.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 4.10nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 3nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in human urotensin-2-mediated aortic ring contr...More data for this Ligand-Target Pair
Affinity DataEC50: 13nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 8.5nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 9.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 6.30nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 4.90nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 3.70nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 4nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 5.80nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 5.20nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 6.60nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 3.5nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 18nMAssay Description:Allosteric modulation of urotensin-2 receptor in Sprague-Dawley rat thoracic aorta assessed as change in URP-mediated aortic ring contraction by meas...More data for this Ligand-Target Pair
Affinity DataEC50: 117nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced G12 activation by measuring URP pEC50...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+3nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced G12 activation by measuring URP pEC50...More data for this Ligand-Target Pair
Affinity DataEC50: 1.95E+3nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced G12 activation by measuring URP pEC50...More data for this Ligand-Target Pair
Affinity DataEC50: 8.5nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced Gq activation by measur...More data for this Ligand-Target Pair
Affinity DataEC50: 14nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced Gq activation by measur...More data for this Ligand-Target Pair
Affinity DataEC50: 11nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced Gq activation by measur...More data for this Ligand-Target Pair
Affinity DataEC50: 7.10nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced Gq activation by measuring URP pEC50 ...More data for this Ligand-Target Pair
Affinity DataEC50: 4.20nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced Gq activation by measuring URP pEC50 ...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in URP-induced Gq activation by measuring URP pEC50 ...More data for this Ligand-Target Pair
Affinity DataEC50: 2.19E+3nMAssay Description:Allosteric modulation of human urotensin-2 receptor expressed in HEK293 cells assessed as change in human urotensin-2-induced G12 activation by measu...More data for this Ligand-Target Pair
