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Found 6 Enz. Inhib. hit(s) with all data for entry = 50002029
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50452450(CHEMBL4211565)
Affinity DataIC50:  2.97E+3nMAssay Description:Inhibition of recombinant human GST-tagged PDK1 expressed in baculovirus infected Sf9 cells using PDHA1 as substrate measured after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50452449(CHEMBL4218938)
Affinity DataIC50:  3.14E+3nMAssay Description:Inhibition of recombinant human GST-tagged PDK1 expressed in baculovirus infected Sf9 cells using PDHA1 as substrate measured after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50452450(CHEMBL4211565)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of recombinant human GST-tagged PDK2 expressed in baculovirus infected Sf9 cells using PDHA1 as substrate measured after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM50452449(CHEMBL4218938)
Affinity DataIC50:  1.09E+4nMAssay Description:Inhibition of recombinant human GST-tagged PDK2 expressed in baculovirus infected Sf9 cells using PDHA1 as substrate measured after 1 hr by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 1, mitochondrial(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM227588(DCA)
Affinity DataIC50:  5.10E+6nMAssay Description:Inhibition of recombinant human GST-tagged PDK1 expressed in baculovirus infected Sf9 cells using PDHA1 as substrate measured after 1 hr by ELISAMore data for this Ligand-Target Pair
Target[Pyruvate dehydrogenase (acetyl-transferring)] kinase isozyme 2, mitochondrial(Homo sapiens (Human))
Sichuan University

Curated by ChEMBL
LigandPNGBDBM227588(DCA)
Affinity DataIC50:  9.00E+6nMAssay Description:Inhibition of recombinant human GST-tagged PDK2 expressed in baculovirus infected Sf9 cells using PDHA1 as substrate measured after 1 hr by ELISAMore data for this Ligand-Target Pair