Found 28 Enz. Inhib. hit(s) with all data for entry = 50001456 
Affinity DataIC50: 0.200nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by in cell western assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by in cell western assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by in cell western assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by in cell western assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Competitive inhibition against rat cytoplasmic Thymidine kinaseMore data for this Ligand-Target Pair
Affinity DataIC50: 0.700nMAssay Description:Ability to inhibit the rat muscle adenylate kinase lII in competition with the AMP variedMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) expressed in Escherichia coli assessed as inhibition of estrad...More data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 3nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) Y537S mutant expressed in Escherichia coli assessed as inhibit...More data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 4nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) D538G mutant expressed in Escherichia coli assessed as inhibit...More data for this Ligand-Target Pair
Affinity DataIC50: 11nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 12nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 16nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) D538G mutant expressed in Escherichia coli assessed as inhibit...More data for this Ligand-Target Pair
Affinity DataIC50: 18nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Ability to inhibit the rat muscle adenylate kinase lII in competition with the AMP variedMore data for this Ligand-Target Pair
Affinity DataIC50: 29nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) Y537S mutant expressed in Escherichia coli assessed as inhibit...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Induction of ERalpha degradation in human MCF7 cells after 4 hrs by in cell western assayMore data for this Ligand-Target Pair
Affinity DataIC50: 47nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 50nMAssay Description:Ability to inhibit the rat muscle adenylate kinase(AK II) isozyme in competition with the AMP variedMore data for this Ligand-Target Pair
Affinity DataIC50: 67nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) Y537S mutant expressed in Escherichia coli assessed as inhibit...More data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Beta-2 adrenergic receptor antagonistic activity on guinea pig tracheal chainsMore data for this Ligand-Target Pair
Affinity DataIC50: 284nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) expressed in Escherichia coli assessed as inhibition of estrad...More data for this Ligand-Target Pair
Affinity DataIC50: 728nMAssay Description:Antagonist activity at recombinant human His6-tagged ERalpha LBD (298 to 554 residues) Y537S mutant expressed in Escherichia coli assessed as inhibit...More data for this Ligand-Target Pair
Affinity DataIC50: 937nMAssay Description:Ability to inhibit the rat muscle adenylate kinase (AK II) isozyme in competition with the AMP variedMore data for this Ligand-Target Pair
