Compile Data Set for Download or QSAR
maximum 50k data
Found 50 Enz. Inhib. hit(s) with all data for entry = 50002557
TargetGlucagon-like peptide 1 receptor(Mus musculus)
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459979(CHEMBL4227636)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at mouse GLP1 receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459983(CHEMBL4224701)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459981(CHEMBL4225594)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  41nMAssay Description:Agonist activity at human GLP1 receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459979(CHEMBL4227636)
Affinity DataEC50:  0.0900nMAssay Description:Agonist activity at human GLP1 receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at mouse GCG receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459980(CHEMBL4227861)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459982(CHEMBL4226514)
Affinity DataEC50:  0.0150nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459983(CHEMBL4224701)
Affinity DataEC50:  0.0680nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459984(CHEMBL4225795)
Affinity DataEC50:  0.00300nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459985(CHEMBL4226451)
Affinity DataEC50:  0.115nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459986(CHEMBL4226634)
Affinity DataEC50:  0.00400nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459987(CHEMBL4226613)
Affinity DataEC50:  0.0310nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459988(CHEMBL4227045)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459989(CHEMBL4225340)
Affinity DataEC50:  0.0410nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459984(CHEMBL4225795)
Affinity DataEC50:  0.00600nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459990(CHEMBL4224968)
Affinity DataEC50:  0.00500nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459991(CHEMBL4226185)
Affinity DataEC50:  0.00900nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459992(CHEMBL4227180)
Affinity DataEC50:  0.00400nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459981(CHEMBL4225594)
Affinity DataEC50:  0.867nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459988(CHEMBL4227045)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459989(CHEMBL4225340)
Affinity DataEC50:  2.70nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459984(CHEMBL4225795)
Affinity DataEC50:  1.70nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459990(CHEMBL4224968)
Affinity DataEC50:  1.10nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459985(CHEMBL4226451)
Affinity DataEC50:  5.80nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459986(CHEMBL4226634)
Affinity DataEC50:  0.133nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459989(CHEMBL4225340)
Affinity DataEC50:  0.0390nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459992(CHEMBL4227180)
Affinity DataEC50:  0.00200nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459982(CHEMBL4226514)
Affinity DataEC50:  0.0280nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459982(CHEMBL4226514)
Affinity DataEC50:  2.20nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459992(CHEMBL4227180)
Affinity DataEC50:  0.812nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  0.5nMAssay Description:Agonist activity at human GCG receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Mus musculus)
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459979(CHEMBL4227636)
Affinity DataEC50: >100nMAssay Description:Agonist activity at mouse GCG receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459990(CHEMBL4224968)
Affinity DataEC50:  0.0930nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459993(CHEMBL4229251)
Affinity DataEC50:  0.00300nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459993(CHEMBL4229251)
Affinity DataEC50:  3.5nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459987(CHEMBL4226613)
Affinity DataEC50:  0.0220nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459986(CHEMBL4226634)
Affinity DataEC50:  0.00700nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459981(CHEMBL4225594)
Affinity DataEC50:  5.20nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459988(CHEMBL4227045)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459979(CHEMBL4227636)
Affinity DataEC50: >1.00E+3nMAssay Description:Agonist activity at human GCG receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Mus musculus)
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50266693(CHEBI:5391 | Glucagen Hypokit | Glucagon | Glucago...)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at mouse GLP1 receptor expressed in CHO cells assessed as increase in cAMP level by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459993(CHEMBL4229251)
Affinity DataEC50:  0.00300nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon-like peptide 1 receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459991(CHEMBL4226185)
Affinity DataEC50:  0.0400nMAssay Description:Agonist activity at human GLP1 receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter ge...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459980(CHEMBL4227861)
Affinity DataEC50:  0.150nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGlucagon receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459985(CHEMBL4226451)
Affinity DataEC50:  0.0160nMAssay Description:Agonist activity at human GCG receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459987(CHEMBL4226613)
Affinity DataEC50:  6.30nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459983(CHEMBL4224701)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459991(CHEMBL4226185)
Affinity DataEC50:  1.60nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGastric inhibitory polypeptide receptor(Homo sapiens (Human))
Novo Nordisk Research Center Indianapolis

Curated by ChEMBL
LigandPNGBDBM50459980(CHEMBL4227861)
Affinity DataEC50:  5.5nMAssay Description:Agonist activity at human GIP receptor expressed in HEK293 cells assessed as increase in cAMP level after 5 hrs by CRE driven luciferase reporter gen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed