Compile Data Set for Download or QSAR
Report error Found 12 Enz. Inhib. hit(s) with all data for entry = 50002043
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452620(CHEMBL4218860)
Affinity DataIC50: 1.20E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452625(CHEMBL4208818)
Affinity DataIC50: 1.23E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452629(CHEMBL4204474)
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452627(CHEMBL4208352)
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 1.46E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452626(CHEMBL4204616)
Affinity DataIC50: 2.71E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452628(CHEMBL4212660)
Affinity DataIC50: 3.44E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452619(CHEMBL4211314)
Affinity DataIC50: 3.89E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452617(CHEMBL4207420)
Affinity DataIC50: 4.06E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452621(CHEMBL4205810)
Affinity DataIC50: 4.33E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452618(CHEMBL4217801)
Affinity DataIC50: 4.88E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetAcetylcholinesterase(Mouse)
Panjab University

Curated by ChEMBL
LigandPNGBDBM50452624(CHEMBL4212031)
Affinity DataIC50: 7.97E+4nMAssay Description:Inhibition of AchE in albino LACA mouse brain using acetylthiocholine iodide as substrate incubated for 10 mins measured for 2 mins by Ellman's metho...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed