Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50001555
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284915(CHEMBL4169808)
Affinity DataIC50:  14nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284923(CHEMBL4171996)
Affinity DataIC50:  32nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284942(CHEMBL4163704)
Affinity DataIC50:  36nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM13061(4,4 -(1H-1,2,4-triazol-1-ylmethanediyl)dibenzonitr...)
Affinity DataIC50:  50nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284913(CHEMBL4175438)
Affinity DataIC50:  51nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50285027(CHEMBL4176600)
Affinity DataIC50:  54nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50285026(CHEMBL4162931)
Affinity DataIC50:  58nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284941(CHEMBL4167569)
Affinity DataIC50:  83nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284939(CHEMBL4161492)
Affinity DataIC50:  97nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284946(CHEMBL4160335)
Affinity DataIC50:  109nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50285029(CHEMBL4159159)
Affinity DataIC50:  197nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284981(CHEMBL4169419)
Affinity DataIC50:  208nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284947(CHEMBL4161789)
Affinity DataIC50:  211nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284980(CHEMBL4165988)
Affinity DataIC50:  217nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50285004(CHEMBL4173231)
Affinity DataIC50:  238nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50285030(CHEMBL4164126)
Affinity DataIC50:  261nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284943(CHEMBL4174373)
Affinity DataIC50:  277nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284940(CHEMBL4170868)
Affinity DataIC50:  677nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284938(CHEMBL4170941)
Affinity DataIC50:  1.06E+3nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50284912(CHEMBL4172433)
Affinity DataIC50:  2.64E+3nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAromatase(Homo sapiens (Human))
Yunnan University

Curated by ChEMBL
LigandPNGBDBM50285028(CHEMBL4162549)
Affinity DataIC50:  7.77E+3nMAssay Description:Inhibition of human aromatase using androstenedione as substrate and NADPH preincubated for 24 hrs followed by substrate addition measured after 24 h...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed