BindingDB PrimarySearch_ki

Found 42 Enz. Inhib. hit(s) with all data for entry = 50002144

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)

Ki: 3.70nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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3D Structure (crystal)

Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)

Ki: 29nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454107(CHEMBL4218702)

Ki: 45nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454105(CHEMBL4205229)

Ki: 73nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454100(CHEMBL4206866)

Ki: 76nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454102(CHEMBL4208621)

Ki: 247nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454098(CHEMBL4207394)

Ki: 609nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454112(CHEMBL4211237)

Ki: 708nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454106(CHEMBL4214129)

Ki: 724nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454097(CHEMBL4215999)

Ki: 800nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454108(CHEMBL4204923)

Ki: 857nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454095(CHEMBL4202505)

Ki: 1.19E+3nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454101(CHEMBL4211754)

Ki: 1.25E+3nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454104(CHEMBL4216812)

Ki: 1.29E+3nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454096(CHEMBL4210184)

Ki: 1.46E+3nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454095(CHEMBL4202505)

Ki: 2.55E+3nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454103(CHEMBL4213942)

Ki: 3.60E+3nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454111(CHEMBL4211647)

Ki: >1.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454110(CHEMBL4203335)

Ki: >1.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454109(CHEMBL4202650)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454111(CHEMBL4211647)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454103(CHEMBL4213942)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454102(CHEMBL4208621)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454112(CHEMBL4211237)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454105(CHEMBL4205229)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454110(CHEMBL4203335)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454097(CHEMBL4215999)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454109(CHEMBL4202650)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454108(CHEMBL4204923)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454100(CHEMBL4206866)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454107(CHEMBL4218702)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454106(CHEMBL4214129)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454098(CHEMBL4207394)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
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Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454099(CHEMBL4216317)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454099(CHEMBL4216317)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB1 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454104(CHEMBL4216812)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454096(CHEMBL4210184)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 2(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454101(CHEMBL4211754)

Ki: >4.00E+4nMAssay Description:Displacement of [3H]CP,55-940 from recombinant human CB2 receptor expressed in HEK293 EBNA cell membranes after 90 mins by microbeta scintillation co...More data for this Ligand-Target Pair

PDB Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)

IC50: 9.70nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHO cell membranes assessed as reduction in GTPgammaS binding after 30 mins by microbeta count...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

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Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454100(CHEMBL4206866)

IC50: 182nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHO cell membranes assessed as reduction in GTPgammaS binding after 30 mins by microbeta count...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454107(CHEMBL4218702)

IC50: 249nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHO cell membranes assessed as reduction in GTPgammaS binding after 30 mins by microbeta count...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed

Cannabinoid receptor 1(Homo sapiens (Human))
University Of Sassari

Curated by ChEMBL

PNG

BDBM50454105(CHEMBL4205229)

IC50: 550nMAssay Description:Antagonist activity at human CB1 receptor expressed in CHO cell membranes assessed as reduction in GTPgammaS binding after 30 mins by microbeta count...More data for this Ligand-Target Pair

PDB NCI pathway Reactome pathway KEGG
UniProtKB/SwissProt
DrugBank antibodypedia GoogleScholar

Details Article PubMed