TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomesMore data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 430nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of mPGES1 (unknown origin) assessed as reduction in conversion of PGH to PGE2More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 1.15E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 1.80E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomesMore data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 2.10E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of ovine COX1 using arachidonic acid as substrate pretreated for 5 mins followed by substrate addition and measured after 5 mins by HPLC a...More data for this Ligand-Target Pair
TargetProstaglandin E synthase(Homo sapiens (Human))
Abdul Wali Khan University Mardan
Curated by ChEMBL
Abdul Wali Khan University Mardan
Curated by ChEMBL
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of mPGES1 in human A549 cell microsomal membrane using pGH2 as substrate pretreated for 15 mins followed by substrate addition and measure...More data for this Ligand-Target Pair