Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50002936
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464950BDBM50464950(CHEMBL4277084)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464954BDBM50464954(CHEMBL4290458)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464949BDBM50464949(CHEMBL4288827)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464952BDBM50464952(CHEMBL4290873)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464957BDBM50464957(CHEMBL4291770)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464948BDBM50464948(CHEMBL4069395)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464956BDBM50464956(CHEMBL4280239)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464951BDBM50464951(CHEMBL4294266)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464953BDBM50464953(CHEMBL4282585)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPotassium voltage-gated channel subfamily H member 2(Human)
Sapienza University of Rome

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50464955BDBM50464955(CHEMBL4292234)
Affinity DataIC50: 5.00E+4nMAssay Description:Inhibition of human ERG by [3H]dofetilide binding displacement assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed