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Found 27 Enz. Inhib. hit(s) with all data for entry = 50002174
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454579(CHEMBL4215648)
Affinity DataIC50:  900nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454590(CHEMBL4207363)
Affinity DataIC50:  1.17E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454578(CHEMBL4203014)
Affinity DataIC50:  1.67E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454591(CHEMBL4205662)
Affinity DataIC50:  1.84E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454576(CHEMBL4202481)
Affinity DataIC50:  1.86E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454572(CHEMBL4218927)
Affinity DataIC50:  2.31E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454589(CHEMBL4218412)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454593(CHEMBL4214007)
Affinity DataIC50:  2.42E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454569(CHEMBL4216922)
Affinity DataIC50:  2.82E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454587(CHEMBL2440274)
Affinity DataIC50:  2.98E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454566(CHEMBL4203968)
Affinity DataIC50:  3.19E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454581(CHEMBL4205472)
Affinity DataIC50:  3.55E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 9.8 nM human tPA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454594(CHEMBL4210355)
Affinity DataIC50:  3.56E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 9.8 nM human tPA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454586(CHEMBL4206843)
Affinity DataIC50:  3.63E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454585(CHEMBL4206161)
Affinity DataIC50:  4.11E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454583(CHEMBL4205996)
Affinity DataIC50:  4.74E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 9.8 nM human tPA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454571(CHEMBL4214513)
Affinity DataIC50:  5.20E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454588(CHEMBL4209604)
Affinity DataIC50:  5.52E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454574(CHEMBL4211050)
Affinity DataIC50:  6.41E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454584(CHEMBL4218241)
Affinity DataIC50:  7.39E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 9.8 nM human tPA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454582(CHEMBL4206636)
Affinity DataIC50:  7.45E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 9.8 nM human tPA...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454575(CHEMBL4208644)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454580(CHEMBL4216092)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 9.8 nM human tPA...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454592(CHEMBL4210774)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454570(CHEMBL4213580)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454573(CHEMBL4206674)
Affinity DataIC50:  2.16E+4nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen activator inhibitor 1(Homo sapiens (Human))
Hamari Chemicals

Curated by ChEMBL
LigandPNGBDBM50454577(CHEMBL4211726)
Affinity DataIC50: >4.00E+4nMAssay Description:Inhibition of human PAI-1 assessed as remaining enzyme activity by measuring p-nitroaniline release pre-incubated for 15 mins before 2 nM Spectrozyme...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed