Compile Data Set for Download or QSAR
Report error Found 28 Enz. Inhib. hit(s) with all data for entry = 50002177
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM16285(2-({6-[(3R)-3-aminopiperidin-1-yl]-3-methyl-2,4-di...)
Affinity DataIC50: 4nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454656(CHEMBL4205581)
Affinity DataIC50: 49nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454650(CHEMBL4204176)
Affinity DataIC50: 80nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454653(CHEMBL4212894)
Affinity DataIC50: 400nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454658(CHEMBL4213950)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454649(CHEMBL4215849)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454652(CHEMBL4207996)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454657(CHEMBL4208513)
Affinity DataIC50: 2.50E+3nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454663(CHEMBL4216792)
Affinity DataIC50: 1.04E+4nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454660(CHEMBL4212367)
Affinity DataIC50: 1.15E+4nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454659(CHEMBL4217326)
Affinity DataIC50: 1.72E+4nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454662(CHEMBL4210635)
Affinity DataIC50: 2.15E+4nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454661(CHEMBL4203639)
Affinity DataIC50: 4.65E+4nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 4(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454664(CHEMBL4205100)
Affinity DataIC50: 5.99E+4nMAssay Description:Inhibition of human DPP4 using A-P-7-amido-4-trifluoromethylcoumarin as substrate pretreated for 10 mins followed by substrate addition measured afte...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454650(CHEMBL4204176)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP9 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454649(CHEMBL4215849)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP8 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454649(CHEMBL4215849)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP9 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454652(CHEMBL4207996)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP9 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454653(CHEMBL4212894)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP9 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454650(CHEMBL4204176)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP8 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454657(CHEMBL4208513)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP9 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454652(CHEMBL4207996)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP8 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454658(CHEMBL4213950)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP9 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 9(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454656(CHEMBL4205581)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP9 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454658(CHEMBL4213950)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP8 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454657(CHEMBL4208513)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP8 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454653(CHEMBL4212894)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP8 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetDipeptidyl peptidase 8(Human)
Shanghai Jiao Tong University

Curated by ChEMBL
LigandPNGBDBM50454656(CHEMBL4205581)
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of recombinant human DPP8 using H-Gly-Pro-AMC as substrate measured after 10 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed