Compile Data Set for Download or QSAR
maximum 50k data
Found 6 Enz. Inhib. hit(s) with all data for entry = 50001449
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
Institute For Research In Cancer And Allied Diseases

Curated by ChEMBL
LigandPNGBDBM50280395(CHEMBL4171480)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of recombinant human GST-tagged EPAC1 (149 to 881 residues) expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRap guanine nucleotide exchange factor 4(Homo sapiens (Human))
Institute For Research In Cancer And Allied Diseases

Curated by ChEMBL
LigandPNGBDBM50280396(CHEMBL4160863)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPAC2 expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine nucleotide exchange ac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
Institute For Research In Cancer And Allied Diseases

Curated by ChEMBL
LigandPNGBDBM50280394(CHEMBL4168137)
Affinity DataIC50:  1.76E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPAC1 (149 to 881 residues) expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRap guanine nucleotide exchange factor 4(Homo sapiens (Human))
Institute For Research In Cancer And Allied Diseases

Curated by ChEMBL
LigandPNGBDBM50280395(CHEMBL4171480)
Affinity DataIC50:  2.23E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPAC2 expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine nucleotide exchange ac...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
Institute For Research In Cancer And Allied Diseases

Curated by ChEMBL
LigandPNGBDBM50280396(CHEMBL4160863)
Affinity DataIC50:  3.13E+4nMAssay Description:Inhibition of recombinant human GST-tagged EPAC1 (149 to 881 residues) expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetRap guanine nucleotide exchange factor 3(Homo sapiens (Human))
Institute For Research In Cancer And Allied Diseases

Curated by ChEMBL
LigandPNGBDBM50280397(CHEMBL4175985)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of recombinant human GST-tagged EPAC1 (149 to 881 residues) expressed in Escherichia coli Rosetta 2(DE3) assessed as reduction in guanine ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed