Compile Data Set for Download or QSAR
Report error Found 46 Enz. Inhib. hit(s) with all data for entry = 50002182
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454733BDBM50454733(CHEMBL4204093)
Affinity DataIC50: 1.80nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454731BDBM50454731(CHEMBL4208618)
Affinity DataIC50: 3.60nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454751BDBM50454751(CHEMBL4212160)
Affinity DataIC50: 3.80nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454739BDBM50454739(CHEMBL4205777)
Affinity DataIC50: 4.5nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454774BDBM50454774(CHEMBL4216611)
Affinity DataIC50: 4.80nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454769BDBM50454769(CHEMBL4205893)
Affinity DataIC50: 5.5nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454760BDBM50454760(CHEMBL4202790)
Affinity DataIC50: 5.80nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454724BDBM50454724(CHEMBL4213886)
Affinity DataIC50: 6.20nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454742BDBM50454742(CHEMBL4206718)
Affinity DataIC50: 7nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454732BDBM50454732(CHEMBL4204419)
Affinity DataIC50: 7.40nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454752BDBM50454752(CHEMBL4213750)
Affinity DataIC50: 7.5nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454763BDBM50454763(CHEMBL4206893)
Affinity DataIC50: 7.70nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454741BDBM50454741(CHEMBL4216476)
Affinity DataIC50: 7.80nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454737BDBM50454737(CHEMBL4215483)
Affinity DataIC50: 8.5nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454773BDBM50454773(CHEMBL4217140)
Affinity DataIC50: 8.60nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454734BDBM50454734(CHEMBL4203546)
Affinity DataIC50: 8.70nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454747BDBM50454747(CHEMBL4215626)
Affinity DataIC50: 9nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454735BDBM50454735(CHEMBL4218344)
Affinity DataIC50: 9.40nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454754BDBM50454754(CHEMBL4213555)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454728BDBM50454728(CHEMBL4214577)
Affinity DataIC50: 9.90nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454740BDBM50454740(CHEMBL4205854)
Affinity DataIC50: 10nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454746BDBM50454746(CHEMBL4207248)
Affinity DataIC50: 11nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454736BDBM50454736(CHEMBL4212913)
Affinity DataIC50: 12nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454726BDBM50454726(CHEMBL4215098)
Affinity DataIC50: 12nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454767BDBM50454767(CHEMBL4206681)
Affinity DataIC50: 12nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454749BDBM50454749(CHEMBL4209874)
Affinity DataIC50: 13nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454762BDBM50454762(CHEMBL4208430)
Affinity DataIC50: 13nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454770BDBM50454770(CHEMBL4213636)
Affinity DataIC50: 15nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454738BDBM50454738(CHEMBL4207817)
Affinity DataIC50: 16nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454768BDBM50454768(CHEMBL4204845)
Affinity DataIC50: 16nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454750BDBM50454750(CHEMBL4218341)
Affinity DataIC50: 17nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454727BDBM50454727(CHEMBL4216695)
Affinity DataIC50: 17nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454764BDBM50454764(CHEMBL4202728)
Affinity DataIC50: 17nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454729BDBM50454729(CHEMBL4214390)
Affinity DataIC50: 18nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454745BDBM50454745(CHEMBL4202896)
Affinity DataIC50: 19nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454766BDBM50454766(CHEMBL4203358)
Affinity DataIC50: 22nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454753BDBM50454753(CHEMBL4209292)
Affinity DataIC50: 24nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454761BDBM50454761(CHEMBL4207627)
Affinity DataIC50: 31nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454744BDBM50454744(CHEMBL4202459)
Affinity DataIC50: 35nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454748BDBM50454748(CHEMBL4203427)
Affinity DataIC50: 40nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454725BDBM50454725(CHEMBL4212704)
Affinity DataIC50: 49nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454743BDBM50454743(CHEMBL4209873)
Affinity DataIC50: 51nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454771BDBM50454771(CHEMBL4207782)
Affinity DataIC50: 54nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454772BDBM50454772(CHEMBL4210669)
Affinity DataIC50: 67nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454730BDBM50454730(CHEMBL4212129)
Affinity DataIC50: 90nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetGlutaminyl-peptide cyclotransferase(Human)
Seoul National University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454765BDBM50454765(CHEMBL4214145)
Affinity DataIC50: 117nMAssay Description:Inhibition of human glutaminyl cyclase using Gln-AMC as substrate by pGAPase coupled fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed