Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50002186
TargetLipopolysaccharide heptosyltransferase 1(Escherichia coli (strain K12))
Wesleyan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 34103BDBM34103(dextrose | glucose | D-glucose)
Affinity DataKi:  2.80E+5nMAssay Description:Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetLipopolysaccharide heptosyltransferase 1(Escherichia coli (strain K12))
Wesleyan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454776BDBM50454776(CHEMBL4209246)
Affinity DataKi:  3.40E+5nMAssay Description:Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetLipopolysaccharide heptosyltransferase 1(Escherichia coli (strain K12))
Wesleyan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 20876BDBM20876((2R,3S,4S,5R,6S)-2-(hydroxymethyl)-6-methoxyoxane-...)
Affinity DataKi:  3.70E+5nMAssay Description:Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetLipopolysaccharide heptosyltransferase 1(Escherichia coli (strain K12))
Wesleyan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 228805BDBM228805(Galactose)
Affinity DataKi:  5.00E+5nMAssay Description:Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetLipopolysaccharide heptosyltransferase 1(Escherichia coli (strain K12))
Wesleyan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454780BDBM50454780(CHEMBL4212177)
Affinity DataKi:  5.20E+5nMAssay Description:Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetLipopolysaccharide heptosyltransferase 1(Escherichia coli (strain K12))
Wesleyan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454777BDBM50454777(CHEMBL4205643)
Affinity DataKi:  5.70E+5nMAssay Description:Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetLipopolysaccharide heptosyltransferase 1(Escherichia coli (strain K12))
Wesleyan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454779BDBM50454779(CHEMBL4213641)
Affinity DataKi:  6.50E+5nMAssay Description:Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed
TargetLipopolysaccharide heptosyltransferase 1(Escherichia coli (strain K12))
Wesleyan University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50454778BDBM50454778(CHEMBL132186 | CHEBI:320055)
Affinity DataKi:  6.80E+5nMAssay Description:Inhibition of Escherichia coli Heptosyltransferase I assessed as reduction in ADP release using ODLA and ADP-heptose substrates in presence of phosph...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/15/2020
Entry Details Article
PubMed