Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50001707
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Alagappa University

Curated by ChEMBL
LigandPNGBDBM50293760(2-(3-fluoro-4-methoxyphenylamino)-1-(2-(trifluorom...)
Affinity DataIC50:  459nMAssay Description:Inhibition of mitotic kinesin Eg5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Alagappa University

Curated by ChEMBL
LigandPNGBDBM23772((2R)-2-amino-3-[(triphenylmethyl)sulfanyl]propanoi...)
Affinity DataIC50:  1.00E+3nMAssay Description:Inhibition of mitotic kinesin Eg5 (unknown origin)More data for this Ligand-Target Pair
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Alagappa University

Curated by ChEMBL
LigandPNGBDBM50316145(CHEMBL4176343)
Affinity DataIC50:  4.86E+3nMAssay Description:Inhibition of human mitotic kinesin Eg5 motor domain (1 to 368 residues) assessed as reduction in steady-state basal ATPase activity using ATP as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Alagappa University

Curated by ChEMBL
LigandPNGBDBM50316143(CHEMBL4159757)
Affinity DataIC50:  9.03E+3nMAssay Description:Inhibition of human mitotic kinesin Eg5 motor domain (1 to 368 residues) assessed as reduction in steady-state basal ATPase activity using ATP as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin-like protein KIF11(Homo sapiens (Human))
Alagappa University

Curated by ChEMBL
LigandPNGBDBM50316144(CHEMBL4166354)
Affinity DataIC50:  1.14E+4nMAssay Description:Inhibition of human mitotic kinesin Eg5 motor domain (1 to 368 residues) assessed as reduction in steady-state basal ATPase activity using ATP as sub...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed