TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California-Riverside
Curated by ChEMBL
University Of California-Riverside
Curated by ChEMBL
Affinity DataIC50: 5.20nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly26 residues) expressed in Escherichia coli BL21 codon plus using Mca-Pro-Leu-Gly...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California-Riverside
Curated by ChEMBL
University Of California-Riverside
Curated by ChEMBL
Affinity DataIC50: 55nMAssay Description:Inhibition of recombinant human MMP12 catalytic domain (Gly106 to Gly26 residues) expressed in Escherichia coli BL21 codon plus using Mca-Pro-Leu-Gly...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California-Riverside
Curated by ChEMBL
University Of California-Riverside
Curated by ChEMBL
Affinity DataKd: <50nMAssay Description:Binding affinity to recombinant human MMP12 catalytic domain (Gly106 to Gly26 residues) expressed in Escherichia coli BL21 codon plus by 1D 1H alipha...More data for this Ligand-Target Pair
TargetMacrophage metalloelastase(Homo sapiens (Human))
University Of California-Riverside
Curated by ChEMBL
University Of California-Riverside
Curated by ChEMBL
Affinity DataKd: <50nMAssay Description:Binding affinity to recombinant human MMP12 catalytic domain (Gly106 to Gly26 residues) expressed in Escherichia coli BL21 codon plus by 2D [15N,1H] ...More data for this Ligand-Target Pair