Compile Data Set for Download or QSAR
Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50000620
TargetToll-like receptor 4(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255625(CHEMBL4070714)
Affinity DataIC50: 630nMAssay Description:Antagonist activity at human TLR4 expressed in HEK blue cells assessed as inhibition of LPS-induced NF-kappaB activation-mediated SEAP production pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255625(CHEMBL4070714)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at human TLR4 expressed in mouse RAW blue cells assessed as inhibition of LPS-induced NF-kappaB activation-mediated SEAP producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255632(CHEMBL4100044)
Affinity DataIC50: 2.00E+3nMAssay Description:Antagonist activity at human TLR4 expressed in HEK blue cells assessed as inhibition of LPS-induced NF-kappaB activation-mediated SEAP production pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed
TargetLymphocyte antigen 96(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255632(CHEMBL4100044)
Affinity DataKd:  3.00E+3nMAssay Description:Binding to C-terminal His6-tagged human MD2 expressed in Pichia pastoris GS115 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255626(CHEMBL4069693)
Affinity DataIC50: 5.45E+3nMAssay Description:Antagonist activity at human TLR4 expressed in HEK blue cells assessed as inhibition of LPS-induced NF-kappaB activation-mediated SEAP production pre...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255632(CHEMBL4100044)
Affinity DataIC50: 7.70E+3nMAssay Description:Antagonist activity at human TLR4 expressed in mouse RAW blue cells assessed as inhibition of LPS-induced NF-kappaB activation-mediated SEAP producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed
TargetLymphocyte antigen 96(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255625(CHEMBL4070714)
Affinity DataKd:  1.40E+4nMAssay Description:Binding to C-terminal His6-tagged human MD2 expressed in Pichia pastoris GS115 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed
TargetLymphocyte antigen 96(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255626(CHEMBL4069693)
Affinity DataKd:  2.20E+4nMAssay Description:Binding to C-terminal His6-tagged human MD2 expressed in Pichia pastoris GS115 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed
TargetToll-like receptor 4(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255626(CHEMBL4069693)
Affinity DataIC50: 4.20E+4nMAssay Description:Antagonist activity at human TLR4 expressed in mouse RAW blue cells assessed as inhibition of LPS-induced NF-kappaB activation-mediated SEAP producti...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed
TargetLymphocyte antigen 96(Human)
University of Milano-Bicocca

Curated by ChEMBL
LigandPNGBDBM50255633(CHEMBL4091601)
Affinity DataKd:  6.70E+4nMAssay Description:Binding to C-terminal His6-tagged human MD2 expressed in Pichia pastoris GS115 by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/15/2019
Entry Details Article
PubMed