Compile Data Set for Download or QSAR
Report error Found 55 Enz. Inhib. hit(s) with all data for entry = 50014380
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575379BDBM50575379(CHEMBL4852814)
Affinity DataIC50: 150nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575376BDBM50575376(CHEMBL4854119)
Affinity DataIC50: 200nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575413BDBM50575413(CHEMBL4877679)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575384BDBM50575384(CHEMBL4866473)
Affinity DataIC50: 300nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575404BDBM50575404(CHEMBL4863558)
Affinity DataIC50: 400nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575409BDBM50575409(CHEMBL4863725)
Affinity DataIC50: 400nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575378BDBM50575378(CHEMBL4849241)
Affinity DataIC50: 400nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575377BDBM50575377(CHEMBL4874714)
Affinity DataIC50: 500nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575383BDBM50575383(CHEMBL4849781)
Affinity DataIC50: 500nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575387BDBM50575387(CHEMBL4848036)
Affinity DataIC50: 500nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575382BDBM50575382(CHEMBL4864461)
Affinity DataIC50: 600nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575386BDBM50575386(CHEMBL4852450)
Affinity DataIC50: 700nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575385BDBM50575385(CHEMBL4877290)
Affinity DataIC50: 750nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575405BDBM50575405(CHEMBL4848692)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 1(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575413BDBM50575413(CHEMBL4877679)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat UT-B incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575403BDBM50575403(CHEMBL4877908)
Affinity DataIC50: 800nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575417BDBM50575417(CHEMBL4875031)
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575399BDBM50575399(CHEMBL4849280)
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575408BDBM50575408(CHEMBL4859014)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575411BDBM50575411(CHEMBL4861819)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575381BDBM50575381(CHEMBL4856839)
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575407BDBM50575407(CHEMBL4867965)
Affinity DataIC50: 1.40E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575380BDBM50575380(CHEMBL4852161)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575412BDBM50575412(CHEMBL4866447)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575398BDBM50575398(CHEMBL4866155)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575415BDBM50575415(CHEMBL4864170)
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 1(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575379BDBM50575379(CHEMBL4852814)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat UT-B incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 41258BDBM41258(SMR000079192 | MLS000065400 | N-(3-isoxazolyl)-2-p...)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575406BDBM50575406(CHEMBL4866180)
Affinity DataIC50: 2.70E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 1(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575416BDBM50575416(CHEMBL4859518)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rat UT-B incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575414BDBM50575414(CHEMBL4878494)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575416BDBM50575416(CHEMBL4859518)
Affinity DataIC50: 3.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 1(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575403BDBM50575403(CHEMBL4877908)
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of rat UT-B incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575396BDBM50575396(CHEMBL4872678)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575418BDBM50575418(CHEMBL4874369)
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575419BDBM50575419(CHEMBL4847861)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 1(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575417BDBM50575417(CHEMBL4875031)
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of rat UT-B incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575395BDBM50575395(CHEMBL4876728)
Affinity DataIC50: 8.00E+3nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 1(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575418BDBM50575418(CHEMBL4874369)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of rat UT-B incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 1(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575419BDBM50575419(CHEMBL4847861)
Affinity DataIC50: 1.40E+4nMAssay Description:Inhibition of rat UT-B incubated for 15 minsMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575388BDBM50575388(CHEMBL4856942)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575389BDBM50575389(CHEMBL4853998)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575390BDBM50575390(CHEMBL4852552)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575391BDBM50575391(CHEMBL4871240)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575392BDBM50575392(CHEMBL4856475)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575393BDBM50575393(CHEMBL4851613)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575410BDBM50575410(CHEMBL4867277)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575394BDBM50575394(CHEMBL4857390)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575397BDBM50575397(CHEMBL4852431)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
TargetUrea transporter 2(Rat)
San Francisco State University

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50575400BDBM50575400(CHEMBL4853194)
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of rat UT-A1 expressed in MDCK cells incubated for 15 mins by fluorescence plate reader assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/23/2022
Entry Details Article
PubMed
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