Compile Data Set for Download or QSAR
maximum 50k data
Found 19 Enz. Inhib. hit(s) with all data for entry = 50002749
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462437(CHEMBL4240338)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462440(CHEMBL4240680)
Affinity DataEC50:  3.86E+4nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50013727(CHEBI:79990 | CHEMBL410478 | GW409544)
Affinity DataEC50:  2.30nMAssay Description:Agonist activity at GAL4-fused human PPARalpha LBDMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462438(CHEMBL4237642)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462439(CHEMBL4237449)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462437(CHEMBL4240338)
Affinity DataEC50:  5.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462439(CHEMBL4237449)
Affinity DataEC50:  5.60E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462437(CHEMBL4240338)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50127222(CHEMBL38508 | GW-0742 | {4-[2-(3-Fluoro-4-trifluor...)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462439(CHEMBL4237449)
Affinity DataEC50: >1.00E+5nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462440(CHEMBL4240680)
Affinity DataEC50:  1.83E+4nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50013727(CHEBI:79990 | CHEMBL410478 | GW409544)
Affinity DataEC50:  0.280nMAssay Description:Agonist activity at GAL4-fused human PPARgamma LBDMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462441(CHEMBL1565327)
Affinity DataEC50:  2.50E+4nMAssay Description:Agonist activity at PPARalpha (unknown origin) expressed in reporter combo cells after 36 hrs by dual luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462441(CHEMBL1565327)
Affinity DataEC50:  5.24E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462440(CHEMBL4240680)
Affinity DataEC50:  2.53E+4nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM28706(2-methyl-2-phenoxypropanoic acid, 25a | 2-methyl-2...)
Affinity DataEC50:  12nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462438(CHEMBL4237642)
Affinity DataEC50:  8.90E+3nMAssay Description:Agonist activity at human PPARdelta after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50030474(Avandamet | Avandaryl | Avandia | BRL-49653 | CHEB...)
Affinity DataEC50:  83nMAssay Description:Agonist activity at human PPARgamma after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
University Of Oklahoma

Curated by ChEMBL
LigandPNGBDBM50462438(CHEMBL4237642)
Affinity DataEC50:  2.10E+3nMAssay Description:Agonist activity at human PPARalpha after 22 to 24 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed