TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 970nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincuba...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.57E+3nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincuba...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.78E+3nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincuba...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 2.62E+3nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincuba...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.64E+3nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincubated f...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 1.38E+4nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincubated f...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 4.82E+4nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincuba...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-4/beta-2(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: 6.25E+4nMAssay Description:Antagonist activity at human alpha4beta2 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincuba...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincubated f...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-3/beta-4(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha3beta4 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincuba...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Homo sapiens (Human))
California Northstate University College Of Medicine
Curated by ChEMBL
California Northstate University College Of Medicine
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Antagonist activity at human alpha7 nAChR expressed in HEK293 cells assessed as inhibition of (+/-)-epibatidine-induced calcium influx preincubated f...More data for this Ligand-Target Pair