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Found 7 Enz. Inhib. hit(s) with all data for entry = 50001202
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50272016(CHEMBL4130153)
Affinity DataIC50:  120nMAssay Description:Inhibition of Escherichia coli DNA gyrase subunit GyrA/GyrB supercoiling activity using relaxed pBR322 DNA incubated for 15 mins by ethidium bromide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50272019(CHEMBL4127152)
Affinity DataIC50:  120nMAssay Description:Inhibition of Escherichia coli DNA gyrase subunit GyrA/GyrB supercoiling activity using relaxed pBR322 DNA incubated for 15 mins by ethidium bromide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50272016(CHEMBL4130153)
Affinity DataIC50:  120nMAssay Description:Inhibition of Escherichia coli DNA gyrase subunit GyrA/GyrB supercoiling activity using relaxed pBR322 DNA incubated for 15 mins by ethidium bromide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50272017(CHEMBL4130314)
Affinity DataIC50:  1.39E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase subunit GyrA/GyrB supercoiling activity using relaxed pBR322 DNA incubated for 15 mins by ethidium bromide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50272010(CHEMBL4126896)
Affinity DataIC50:  2.32E+4nMAssay Description:Inhibition of Escherichia coli DNA gyrase subunit GyrA/GyrB supercoiling activity using relaxed pBR322 DNA incubated for 15 mins by ethidium bromide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50272018(CHEMBL4126743)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Escherichia coli DNA gyrase subunit GyrA/GyrB supercoiling activity using relaxed pBR322 DNA incubated for 15 mins by ethidium bromide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA gyrase subunit A/B(Escherichia coli (strain K12))
University Of Iowa

Curated by ChEMBL
LigandPNGBDBM50272011(CHEMBL4126889)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of Escherichia coli DNA gyrase subunit GyrA/GyrB supercoiling activity using relaxed pBR322 DNA incubated for 15 mins by ethidium bromide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed