Compile Data Set for Download or QSAR
maximum 50k data
Found 5 Enz. Inhib. hit(s) with all data for entry = 50003233
TargetHeat shock factor protein 1(Homo sapiens (Human))
University Of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50468275(CHEMBL4293406)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of recombinant human HSF1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in HSF1 trimer-5-fluorescein labeled HSE interact...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock factor protein 1(Homo sapiens (Human))
University Of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50468275(CHEMBL4293406)
Affinity DataIC50:  1.50E+4nMAssay Description:Inhibition of recombinant human HSF1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in HSF1 trimer-5-fluorescein labeled HSE interact...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock factor protein 1(Homo sapiens (Human))
University Of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50468276(CHEMBL4284740)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of recombinant human HSF1 expressed in Escherichia coli BL21 (DE3) assessed as reduction in HSF1 trimer-5-fluorescein labeled HSE interact...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock factor protein 1(Homo sapiens (Human))
University Of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50468274(CHEMBL4282794)
Affinity DataEC50: >8.00E+3nMAssay Description:Binding affinity to recombinant human HSF1 monomer delta LZ1-3 mutant expressed in Escherichia coli BL21 (DE3) after 15 mins by fluorescence polariza...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHeat shock factor protein 1(Homo sapiens (Human))
University Of California At San Francisco

Curated by ChEMBL
LigandPNGBDBM50468274(CHEMBL4282794)
Affinity DataEC50:  4.50E+3nMAssay Description:Binding affinity to recombinant human HSF1 monomer expressed in Escherichia coli BL21 (DE3) after 15 mins by fluorescence polarization assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed