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Found 14 Enz. Inhib. hit(s) with all data for entry = 50001818
TargetHistone acetyltransferase(Tetrahymena thermophila (strain SB210))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50372747(CHEMBL4161210)
Affinity DataIC50:  500nMAssay Description:Inhibition of tetrahymena GCN5 (48 to 210 residues)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM82909(5-(2-Thiophen-2-yl-acetylamino)-isophthalic acid d...)
Affinity DataIC50:  2.90E+3nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50371146(CHEMBL4168633)
Affinity DataIC50:  6.80E+3nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50372743(CHEMBL4172975)
Affinity DataIC50:  8.60E+3nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50371231(CHEMBL4171987)
Affinity DataIC50:  1.60E+4nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50372745(CHEMBL4160712)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50370968(CHEMBL4159754)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50370981(CHEMBL4175431)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50370931(CHEMBL4162185)
Affinity DataIC50:  3.40E+4nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50372744(CHEMBL4165080)
Affinity DataIC50:  3.47E+4nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50372746(CHEMBL4170095)
Affinity DataIC50:  8.10E+4nMAssay Description:Inhibition of yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) preincubated for 15 mins followed by biotin tagged H3 peptide ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase KAT2A(Homo sapiens (Human))
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50371233(CHEMBL3347571)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of GCN5 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50371146(CHEMBL4168633)
Affinity DataKd:  4.20E+3nMAssay Description:Binding affinity to yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase GCN5(Saccharomyces cerevisiae S288c)
Shanghai University

Curated by ChEMBL
LigandPNGBDBM50372744(CHEMBL4165080)
Affinity DataKd:  2.62E+4nMAssay Description:Binding affinity to yeast GCN5 (99 to 262 residues) expressed in Escherichia coli BL21 (DE3) by SPR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed