Compile Data Set for Download or QSAR
Report error Found 8 Enz. Inhib. hit(s) with all data for entry = 50002980
TargetBile acid receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50465370(CHEMBL4280310)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at FXR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM402340(US10329286, Example 10 | 6-(3-(2-chloro-4-((5- cyc...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at FXR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50465371(CHEMBL4286228)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at FXR (unknown origin) by mammalian one hybrid assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50465371(CHEMBL4286228)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at FXR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM402340(US10329286, Example 10 | 6-(3-(2-chloro-4-((5- cyc...)
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at FXR (unknown origin) by mammalian one hybrid assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50465370(CHEMBL4280310)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at FXR (unknown origin) by mammalian one hybrid assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM402336(US10329286, Example 8 | 6-(3-(2-chloro-4-((5- cycl...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at FXR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetBile acid receptor(Human)
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM402336(US10329286, Example 8 | 6-(3-(2-chloro-4-((5- cycl...)
Affinity DataEC50:  593nMAssay Description:Agonist activity at FXR (unknown origin) by mammalian one hybrid assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed