Compile Data Set for Download or QSAR
maximum 50k data
Found 8 Enz. Inhib. hit(s) with all data for entry = 50002980
TargetBile acid receptor(Homo sapiens (Human))
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50465370(CHEMBL4280310)
Affinity DataEC50:  7.10nMAssay Description:Agonist activity at FXR (unknown origin) by mammalian one hybrid assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM402336(6-(3-(2-chloro-4-((5- cyclopropyl-3-(2,6- dimethox...)
Affinity DataEC50:  593nMAssay Description:Agonist activity at FXR (unknown origin) by mammalian one hybrid assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM402340(6-(3-(2-chloro-4-((5- cyclopropyl-3-(3,5- dichloro...)
Affinity DataEC50:  3.40nMAssay Description:Agonist activity at FXR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50465370(CHEMBL4280310)
Affinity DataEC50:  2.60nMAssay Description:Agonist activity at FXR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50465371(CHEMBL4286228)
Affinity DataEC50:  4.80nMAssay Description:Agonist activity at FXR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM402340(6-(3-(2-chloro-4-((5- cyclopropyl-3-(3,5- dichloro...)
Affinity DataEC50:  6.40nMAssay Description:Agonist activity at FXR (unknown origin) by mammalian one hybrid assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM402336(6-(3-(2-chloro-4-((5- cyclopropyl-3-(2,6- dimethox...)
Affinity DataEC50:  15nMAssay Description:Agonist activity at FXR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetBile acid receptor(Homo sapiens (Human))
Therachem Research Medilab

Curated by ChEMBL
LigandPNGBDBM50465371(CHEMBL4286228)
Affinity DataEC50:  4.5nMAssay Description:Agonist activity at FXR (unknown origin) by mammalian one hybrid assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed