Compile Data Set for Download or QSAR
maximum 50k data
Found 11 Enz. Inhib. hit(s) with all data for entry = 50001829
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404946(CHEMBL4172542)
Affinity DataIC50:  1.12E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404945(CHEMBL4176972)
Affinity DataIC50:  4.39E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404818(CHEMBL4165426)
Affinity DataIC50:  5.09E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404951(CHEMBL4176453)
Affinity DataIC50:  6.75E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404476(CHEMBL4169913)
Affinity DataIC50:  7.06E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404949(CHEMBL4172657)
Affinity DataIC50:  7.27E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404859(CHEMBL4164762)
Affinity DataIC50:  7.28E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404947(CHEMBL4167621)
Affinity DataIC50:  7.31E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404460(CHEMBL4168199)
Affinity DataIC50:  8.20E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404952(CHEMBL4170688)
Affinity DataIC50:  8.21E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 1(Homo sapiens (Human))
Universidad De Le£N

Curated by ChEMBL
LigandPNGBDBM50404950(CHEMBL4165844)
Affinity DataIC50:  8.33E+4nMAssay Description:Inhibition of human Top1B expressed in Top1B deficient Saccharomyces cerevisiae EKY3 assessed as decrease in relaxation of supercoiled pSK DNA preinc...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed