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Found 10 Enz. Inhib. hit(s) with all data for entry = 50001836
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405916(CHEMBL4169245)
Affinity DataIC50:  4.41E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB4 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405914(CHEMBL4162777)
Affinity DataIC50:  5.06E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB4 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405915(CHEMBL4173044)
Affinity DataIC50:  6.40E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB4 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405918(CHEMBL4162362)
Affinity DataIC50:  6.43E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB4 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-4(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405917(CHEMBL4161318)
Affinity DataIC50:  8.05E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB4 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405916(CHEMBL4169245)
Affinity DataIC50:  9.71E+3nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB2 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405915(CHEMBL4173044)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB2 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405914(CHEMBL4162777)
Affinity DataIC50:  1.80E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB2 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405918(CHEMBL4162362)
Affinity DataIC50:  2.54E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB2 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
University Of Salerno

Curated by ChEMBL
LigandPNGBDBM50405917(CHEMBL4161318)
Affinity DataIC50:  3.15E+4nMAssay Description:Inhibition of recombinant human N-terminal GST-His6-fused erbB2 expressed in Sf9 insect cells using poly (Glu, Tyr) 4:1 as substrate after 60 mins in...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed