Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50001837
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405927(CHEMBL4177351)
Affinity DataIC50:  77nMAssay Description:Inhibition of BRD4 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50071106(CHEMBL3410002)
Affinity DataIC50:  140nMAssay Description:Inhibition of BRD4 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50399434(CHEMBL2179387)
Affinity DataIC50:  220nMAssay Description:Inhibition of BRD4 (unknown origin) by Alphascreen assayMore data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405923(CHEMBL4175673)
Affinity DataIC50:  1.02E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405924(CHEMBL4165055)
Affinity DataIC50:  1.43E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405925(CHEMBL4159075)
Affinity DataIC50:  1.55E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405926(CHEMBL4171143)
Affinity DataIC50:  3.02E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50238042(CHEMBL4073350)
Affinity DataIC50:  6.83E+3nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405953(CHEMBL4167326)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405919(CHEMBL4163466)
Affinity DataIC50:  1.27E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405921(CHEMBL4170290)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50406028(CHEMBL4170804)
Affinity DataIC50:  1.33E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50406024(CHEMBL4174139)
Affinity DataIC50:  1.87E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50406023(CHEMBL4165445)
Affinity DataIC50:  2.31E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50406027(CHEMBL4162367)
Affinity DataIC50:  2.75E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50405922(CHEMBL4167407)
Affinity DataIC50:  3.22E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50238043(CHEMBL4100505)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50406026(CHEMBL4169300)
Affinity DataIC50:  4.22E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50406025(CHEMBL4177508)
Affinity DataIC50:  4.73E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50406030(CHEMBL4160166)
Affinity DataIC50:  5.08E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Hebei University

Curated by ChEMBL
LigandPNGBDBM50406022(CHEMBL4172354)
Affinity DataIC50:  6.92E+4nMAssay Description:Inhibition of His-tagged BRD4 bromodomain-1 (unknown origin) expressed in Escherichia coli BL21(DE3) using SGRGK(Ac)-GG-K(Ac)-GLG-K(Ac)-GGA-K(Ac)-RHR...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed