TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 23nMAssay Description:Antagonist activity at C-terminal PK-fused human full length TrkA assessed as inhibition of betaNGF-induced protein binding to Shc1-EA by beta-galact...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataIC50: 26nMAssay Description:Antagonist activity at C-terminal PK-fused human full length TrkA assessed as inhibition of betaNGF-induced protein binding to Shc1-EA by beta-galact...More data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataKd: 32nMAssay Description:Binding affinity to DNA-tagged human partial length TrkA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataKd: 1nMAssay Description:Binding affinity to DNA-tagged human partial length TrkA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
Affinity DataKd: 40nMAssay Description:Binding affinity to DNA-tagged human partial length AURKA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
Affinity DataKd: 5.01E+3nMAssay Description:Binding affinity to DNA-tagged human partial length AURKA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
Affinity DataKd: 25nMAssay Description:Binding affinity to DNA-tagged human partial length AURKA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataKd: 1.60nMAssay Description:Binding affinity to DNA-tagged human partial length TrkA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataKd: 3.20nMAssay Description:Binding affinity to DNA-tagged human partial length TrkA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataKd: 4nMAssay Description:Binding affinity to DNA-tagged human partial length TrkA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
TargetHigh affinity nerve growth factor receptor(Homo sapiens (Human))
Heidelberg University
Curated by ChEMBL
Heidelberg University
Curated by ChEMBL
Affinity DataKd: 2.5nMAssay Description:Binding affinity to DNA-tagged human partial length TrkA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
Affinity DataKd: 0.501nMAssay Description:Binding affinity to DNA-tagged human partial length AURKA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
Affinity DataKd: 100nMAssay Description:Binding affinity to DNA-tagged human partial length AURKA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair
Affinity DataKd: 50nMAssay Description:Binding affinity to DNA-tagged human partial length AURKA expressed in mammalian expression system by qPCR methodMore data for this Ligand-Target Pair