Found 6 Enz. Inhib. hit(s) with all data for entry = 50008584 
Affinity DataKi: 29nMAssay Description:Displacement of [125I]-NDP-alpha-MSH from human MC4R expressed in HEK cell membranes after 1 hr by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 42nMAssay Description:Inhibition of N-terminal His6-tagged KDM4A (1 to 359 residues) (unknown origin) expressed in Escherichia coli BL21(DE3) preincubated for 15 mins foll...More data for this Ligand-Target Pair
TargetATPase family AAA domain-containing protein 2(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataIC50: 166nMAssay Description:Induction of ATAD2 bromodomain (unknown origin) dimerizationMore data for this Ligand-Target Pair
TargetParathyroid hormone/parathyroid hormone-related peptide receptor(Homo sapiens (Human))
Astrazeneca
Curated by ChEMBL
Astrazeneca
Curated by ChEMBL
Affinity DataEC50: 0.130nMAssay Description:Agonist activity at PTH1 receptor (unknown origin) assessed as induction of cAMPMore data for this Ligand-Target Pair
Affinity DataKd: 20nMAssay Description:Binding affinity to human plasma kallikreinMore data for this Ligand-Target Pair
Affinity DataKd: 370nMAssay Description:Inhibition of stonin-2 binding to Eps15 (unknown origin)More data for this Ligand-Target Pair
