Compile Data Set for Download or QSAR
maximum 50k data
Found 31 Enz. Inhib. hit(s) with all data for entry = 50001286
TargetCyclin-dependent kinase 2(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK2 (unknown origin) expressed in baculovirus infected Sf9 insect cells using histone H1 as substrate after 1 hr by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  1nMAssay Description:Inhibition of CDK5 (unknown origin) expressed in baculovirus infected Sf9 insect cells using histone H1 as substrate after 1 hr by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  3nMAssay Description:Inhibition of CDK1 (unknown origin) expressed in baculovirus infected Sf9 insect cells using histone H1 as substrate after 1 hr by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 9(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50139171(Dinaciclib | MK-7965 | SCH-727965 | US11643396, Ex...)
Affinity DataIC50:  4nMAssay Description:Inhibition of CDK9 (unknown origin) expressed in baculovirus infected Sf9 insect cells using histone H1 as substrate after 1 hr by liquid scintillati...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274791(CHEMBL4127826)
Affinity DataIC50:  46nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274802(CHEMBL4125881)
Affinity DataIC50:  54nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 6/G1/S-specific cyclin-D3(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274791(CHEMBL4127826)
Affinity DataIC50:  54nMAssay Description:Inhibition of recombinant human CDK6/cyclin D3 after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCDK-activating kinase assembly factor MAT1/Cyclin-H/Cyclin-dependent kinase 7(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274791(CHEMBL4127826)
Affinity DataIC50:  90nMAssay Description:Inhibition of recombinant human CDK7/cyclin H/MNAT1 after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274842(CHEMBL4130285)
Affinity DataIC50:  151nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274804(CHEMBL4128345)
Affinity DataIC50:  153nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274803(CHEMBL4127944)
Affinity DataIC50:  205nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274850(CHEMBL4126871)
Affinity DataIC50:  206nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274840(CHEMBL4128251)
Affinity DataIC50:  241nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274793(CHEMBL4127110)
Affinity DataIC50:  277nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274790(CHEMBL4125785)
Affinity DataIC50:  277nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 4/G1/S-specific cyclin-D1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274791(CHEMBL4127826)
Affinity DataIC50:  278nMAssay Description:Inhibition of recombinant human CDK4/cyclin D1 after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274794(CHEMBL4127271)
Affinity DataIC50:  280nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274795(CHEMBL4126622)
Affinity DataIC50:  286nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274792(CHEMBL4129339)
Affinity DataIC50:  287nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274796(CHEMBL4130124)
Affinity DataIC50:  288nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274847(CHEMBL4129895)
Affinity DataIC50:  288nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274823(CHEMBL4125887)
Affinity DataIC50:  314nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274818(CHEMBL4126973)
Affinity DataIC50:  378nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274773(CHEMBL4129186)
Affinity DataIC50:  380nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274797(CHEMBL4129227)
Affinity DataIC50:  387nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274851(CHEMBL4125933)
Affinity DataIC50:  399nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274824(CHEMBL4129065)
Affinity DataIC50:  405nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274849(CHEMBL4128562)
Affinity DataIC50:  459nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274822(CHEMBL4125743)
Affinity DataIC50:  474nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274848(CHEMBL4126202)
Affinity DataIC50:  501nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 2/G1/S-specific cyclin-E1(Homo sapiens (Human))
Shihezi University

Curated by ChEMBL
LigandPNGBDBM50274843(CHEMBL4127017)
Affinity DataIC50:  567nMAssay Description:Inhibition of recombinant human CDK2/cyclin E after 40 mins by ADP-Glo reagent based luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed