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Found 22 Enz. Inhib. hit(s) with all data for entry = 50001287
TargetThymidine phosphorylase(Homo sapiens (Human))
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274904(CHEMBL4129617)
Affinity DataIC50:  20nMAssay Description:Inhibition of thymidine phosphorylase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM20079(5-chloro-6-[(2-iminopyrrolidin-1-yl)methyl]-1,2,3,...)
Affinity DataIC50:  35nMAssay Description:Inhibition of human placenta thymidine phosphorylase using [6-3H]dThd as substrate after 5 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274861(CHEMBL4129729)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274882(CHEMBL4129587)
Affinity DataIC50:  6.10E+3nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274865(CHEMBL4125852)
Affinity DataIC50:  9.10E+3nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274863(CHEMBL4126296)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274883(CHEMBL4126143)
Affinity DataIC50:  1.22E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274866(CHEMBL4127084)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274884(CHEMBL4127377)
Affinity DataIC50:  2.45E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274902(CHEMBL4129149)
Affinity DataIC50:  2.93E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274901(CHEMBL4125711)
Affinity DataIC50:  2.94E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274899(CHEMBL4129469)
Affinity DataIC50:  3.35E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274900(CHEMBL4129552)
Affinity DataIC50:  3.52E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Homo sapiens (Human))
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50320723(4-(5-mercapto-1,3,4-oxadiazol-2-yl)phenol | 5-(4-h...)
Affinity DataIC50:  3.82E+4nMAssay Description:Inhibition of thymidine phosphorylase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274881(CHEMBL4127013)
Affinity DataIC50:  3.84E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50134399(1,7-Dihydro-pyrrolo[2,3-d]pyrimidine-2,4-dione | 7...)
Affinity DataIC50:  3.87E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274880(CHEMBL4127521)
Affinity DataIC50:  4.35E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274864(CHEMBL4128092)
Affinity DataIC50:  4.52E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274903(CHEMBL4128440)
Affinity DataIC50:  4.62E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274885(CHEMBL4128771)
Affinity DataIC50:  5.35E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274905(CHEMBL4129801)
Affinity DataIC50:  5.46E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetThymidine phosphorylase(Escherichia coli)
Imam Abdulrahman Bin Faisal University

Curated by ChEMBL
LigandPNGBDBM50274862(CHEMBL4129851)
Affinity DataIC50:  6.42E+4nMAssay Description:Inhibition of Escherichia coli thymidine phosphorylase pretreated for 10 mins followed by substrate addition measured at 10 mins interval for 30 mins...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed