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Found 8 Enz. Inhib. hit(s) with all data for entry = 50008585
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50520631(Ametantrone)
Affinity DataIC50:  30nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50520632(CHEMBL4553471)
Affinity DataIC50:  1.06E+3nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50520634(CHEMBL4575796)
Affinity DataIC50:  1.15E+3nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50520633(CHEMBL4448353)
Affinity DataIC50:  4.34E+3nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-beta(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50520636(CHEMBL4467805)
Affinity DataIC50:  5.25E+3nMAssay Description:Poison activity at recombinant human topoisomerase 2beta using pBR322 plasmid as substrate after 30 mins by ethidium bromide staining based agarose g...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50127140((-)-etoposide | (5S,5aR,8aR,9R)-9-(4-hydroxy-3,5-d...)
Affinity DataIC50:  3.38E+4nMAssay Description:Inhibition of recombinant human topoisomerase 2alpha using supercoiled pNO1 plasmid as substrate after 30 mins by SYBR-GOLD staining based fluorimetr...More data for this Ligand-Target Pair
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50362243(CHEMBL1939412)
Affinity DataIC50:  4.40E+4nMAssay Description:Inhibition of recombinant human topoisomerase 2alpha using supercoiled pNO1 plasmid as substrate after 30 mins by SYBR-GOLD staining based fluorimetr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Shandong University

Curated by ChEMBL
LigandPNGBDBM50520635(CHEMBL4435344)
Affinity DataIC50:  6.50E+4nMAssay Description:Inhibition of recombinant human topoisomerase 2alpha using supercoiled pNO1 plasmid as substrate after 30 mins by SYBR-GOLD staining based fluorimetr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed