Compile Data Set for Download or QSAR
Report error Found 80 Enz. Inhib. hit(s) with all data for entry = 50003247
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468502BDBM50468502(CHEMBL4289527)
Affinity DataIC50: 770nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468553BDBM50468553(CHEMBL4282532)
Affinity DataIC50: 1.70E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468532BDBM50468532(CHEMBL1360726)
Affinity DataKd:  1.80E+3nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468532BDBM50468532(CHEMBL1360726)
Affinity DataIC50: 1.90E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468552BDBM50468552(CHEMBL1591311)
Affinity DataIC50: 2.00E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468537BDBM50468537(CHEMBL4286098)
Affinity DataKd:  2.50E+3nMAssay Description:Binding affinity to N-terminal GST-tagged BRPF1 (unknown origin) expressed in Escherichia coli by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468532BDBM50468532(CHEMBL1360726)
Affinity DataKd:  2.70E+3nMAssay Description:Binding affinity to N-terminal GST-tagged BRPF1 (unknown origin) expressed in Escherichia coli by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468537BDBM50468537(CHEMBL4286098)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468534BDBM50468534(CHEMBL4290403)
Affinity DataIC50: 3.40E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468499BDBM50468499(CHEMBL4291774)
Affinity DataKd:  3.50E+3nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468510BDBM50468510(CHEMBL4280181)
Affinity DataIC50: 3.60E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468533BDBM50468533(CHEMBL4282133)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468514BDBM50468514(CHEMBL4277790)
Affinity DataIC50: 4.40E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468515BDBM50468515(CHEMBL4289326)
Affinity DataIC50: 5.40E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468509BDBM50468509(CHEMBL4295210)
Affinity DataKd:  7.10E+3nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468548BDBM50468548(CHEMBL4284975)
Affinity DataIC50: 8.70E+3nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468502BDBM50468502(CHEMBL4289527)
Affinity DataKd:  9.70E+3nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468503BDBM50468503(CHEMBL4282572)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468505BDBM50468505(CHEMBL4293809)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468525BDBM50468525(CHEMBL4283679)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468539BDBM50468539(CHEMBL4285049)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468526BDBM50468526(CHEMBL4276797)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468527BDBM50468527(CHEMBL4290267)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468508BDBM50468508(CHEMBL4287447)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468524BDBM50468524(CHEMBL4292107)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468538BDBM50468538(CHEMBL4281301)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468531BDBM50468531(CHEMBL4294000)
Affinity DataIC50: 1.01E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468535BDBM50468535(CHEMBL4288350)
Affinity DataIC50: 1.05E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468499BDBM50468499(CHEMBL4291774)
Affinity DataKd:  1.09E+4nMAssay Description:Binding affinity to N-terminal GST-tagged BRPF1 (unknown origin) expressed in Escherichia coli by isothermal titration calorimetryMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468517BDBM50468517(CHEMBL4292834)
Affinity DataIC50: 1.10E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468516BDBM50468516(CHEMBL4285918)
Affinity DataKd:  1.10E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468546BDBM50468546(CHEMBL4276793)
Affinity DataKd:  1.60E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468509BDBM50468509(CHEMBL4295210)
Affinity DataIC50: 1.60E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468511BDBM50468511(CHEMBL4293001)
Affinity DataKd:  1.70E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468517BDBM50468517(CHEMBL4292834)
Affinity DataKd:  1.80E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468519BDBM50468519(CHEMBL4295207)
Affinity DataKd:  1.80E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468501BDBM50468501(CHEMBL4287943)
Affinity DataKd:  1.90E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468529BDBM50468529(CHEMBL1394372)
Affinity DataKd: >2.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468549BDBM50468549(CHEMBL4291772)
Affinity DataKd:  2.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468504BDBM50468504(CHEMBL4291009)
Affinity DataIC50: 2.23E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468530BDBM50468530(CHEMBL4278852)
Affinity DataIC50: 2.36E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468550BDBM50468550(CHEMBL4290863)
Affinity DataIC50: 2.50E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468513BDBM50468513(CHEMBL4280367)
Affinity DataKd: >2.50E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468529BDBM50468529(CHEMBL1394372)
Affinity DataIC50: 2.70E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468499BDBM50468499(CHEMBL4291774)
Affinity DataIC50: 3.06E+4nMAssay Description:Inhibition of recombinant human His-tagged BRPF1 using biotinylated H4(1 to 21)K5/8/12/16Ac peptide as substrate after 30 mins by AlphaScreen assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468515BDBM50468515(CHEMBL4289326)
Affinity DataKd:  3.30E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468521BDBM50468521(CHEMBL4285165)
Affinity DataKd:  3.60E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468520BDBM50468520(CHEMBL4280034)
Affinity DataKd:  4.50E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
TargetPeregrin(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468518BDBM50468518(CHEMBL4284556)
Affinity DataKd: >5.00E+4nMAssay Description:Binding affinity to human partial length BRPF1 (E627 to G740 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargetBromodomain-containing protein 4(Human)
University of Zurich

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50468499BDBM50468499(CHEMBL4291774)
Affinity DataKd: >5.00E+4nMAssay Description:Binding affinity to human partial length BRD4 BD1 (N44 to E168 residues) expressed in Escherichia coli BL21 after 1 hr by BROMOscan assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/18/2020
Entry Details Article
PubMed
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