Compile Data Set for Download or QSAR
maximum 50k data
Found 25 Enz. Inhib. hit(s) with all data for entry = 50001308
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276140(CHEMBL4129995)
Affinity DataIC50:  28nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276143(CHEMBL4128547)
Affinity DataIC50:  2.30E+3nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276143(CHEMBL4128547)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276143(CHEMBL4128547)
Affinity DataIC50:  4.50E+3nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276143(CHEMBL4128547)
Affinity DataIC50:  5.30E+3nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276139(CHEMBL4128509)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276141(CHEMBL4128353)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276145(CHEMBL4128630)
Affinity DataIC50:  2.09E+4nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276139(CHEMBL4128509)
Affinity DataIC50:  3.50E+4nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276139(CHEMBL4128509)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276139(CHEMBL4128509)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human SIRT5 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276140(CHEMBL4129995)
Affinity DataIC50:  9.80E+4nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276140(CHEMBL4129995)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT5 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276140(CHEMBL4129995)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276140(CHEMBL4129995)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276141(CHEMBL4128353)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276139(CHEMBL4128509)
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276142(CHEMBL4129734)
Affinity DataIC50:  2.37E+5nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276141(CHEMBL4128353)
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276142(CHEMBL4129734)
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276142(CHEMBL4129734)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT5 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276142(CHEMBL4129734)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276142(CHEMBL4129734)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276141(CHEMBL4128353)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
School Of Pharmacy

Curated by ChEMBL
LigandPNGBDBM50276141(CHEMBL4128353)
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT5 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed