TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 28nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.30E+3nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.80E+3nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 4.50E+3nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 5.30E+3nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.00E+4nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.09E+4nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 3.50E+4nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human SIRT5 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 9.80E+4nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT5 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >2.00E+5nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-2(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: 2.37E+5nMAssay Description:Inhibition of human N-terminal His6-SUMO-tagged SIRT2 (38 to 356 residues) expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubate...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-1(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >3.00E+5nMAssay Description:Inhibition of human SIRT1 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT5 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-6(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT6 (1 to 294 residues) expressed in Escherichia coli Rosetta (DE3) using H3K9AcWW as substrate preincubated for 15 mins follow...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacetylase sirtuin-3, mitochondrial(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT3 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair
TargetNAD-dependent protein deacylase sirtuin-5, mitochondrial(Homo sapiens (Human))
School Of Pharmacy
Curated by ChEMBL
School Of Pharmacy
Curated by ChEMBL
Affinity DataIC50: >5.00E+5nMAssay Description:Inhibition of human SIRT5 expressed in Escherichia coli BL21 using H3K9AcWW as substrate preincubated for 15 mins followed by substrate addition meas...More data for this Ligand-Target Pair