Report error Found 3304 Enz. Inhib. hit(s) with all data for entry = 50022496
TargetCUGBP Elav-like family member 2(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.0460nMAssay Description:Binding affinity to human CELF2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetDual specificity testis-specific protein kinase 1(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.0860nMAssay Description:Binding affinity to human TESK1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetPlatelet-derived growth factor receptor beta(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.0890nMAssay Description:Binding affinity to human PDGFRB incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.100nMAssay Description:Binding affinity to human SNX2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetEukaryotic translation initiation factor 4B(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.100nMAssay Description:Binding affinity to human EIF4B incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.129nMAssay Description:Binding affinity to human PRKCD incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.132nMAssay Description:Binding affinity to human P4HA1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetRNA cytosine C(5)-methyltransferase NSUN2(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.187nMAssay Description:Binding affinity to human NSUN2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Target28S rRNA (cytosine(4447)-C(5))-methyltransferase(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.204nMAssay Description:Binding affinity to human NOP2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetUncharacterized protein FLJ45252(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.210nMAssay Description:Binding affinity to human FLJ45252 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetSRA stem-loop-interacting RNA-binding protein, mitochondrial(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.214nMAssay Description:Binding affinity to human SLIRP incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetT-complex protein 1 subunit epsilon(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.216nMAssay Description:Binding affinity to human CCT5 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.224nMAssay Description:Binding affinity to human CLK1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetSmall ribosomal subunit protein uS4(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.236nMAssay Description:Binding affinity to human RPS9 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetER lumen protein-retaining receptor 1(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.253nMAssay Description:Binding affinity to human KDELR1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.256nMAssay Description:Binding affinity to human RRP12 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.266nMAssay Description:Binding affinity to human TGFBR1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.296nMAssay Description:Binding affinity to human CDK6 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Nano Luc-fused full length C-terminal EPHA3 (unknown origin) expressed in HEK293T cells using NanoGlo as substrate incubated for 2 hrs ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Nano Luc-fused full length C-terminal EPHA3 (unknown origin) expressed in HEK293T cells using NanoGlo as substrate incubated for 2 hrs ...More data for this Ligand-Target Pair
TargetRNA cytidine acetyltransferase(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.302nMAssay Description:Binding affinity to human NAT10 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetNuclear mitotic apparatus protein 1(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.308nMAssay Description:Binding affinity to human NUMA1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetTelomere length regulation protein TEL2 homolog(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.314nMAssay Description:Binding affinity to human TELO2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetPleckstrin homology domain-containing family G member 3(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.315nMAssay Description:Binding affinity to human PLEKHG3 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetMyosin light chain kinase, smooth muscle(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.317nMAssay Description:Binding affinity to human MYLK incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.337nMAssay Description:Binding affinity to human KIAA0196 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetATP-binding cassette sub-family E member 1(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.362nMAssay Description:Binding affinity to human ABCE1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.373nMAssay Description:Binding affinity to human KDM1A incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetQueuine tRNA-ribosyltransferase accessory subunit 2(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.411nMAssay Description:Binding affinity to human QTRTD1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.443nMAssay Description:Binding affinity to human CUL1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.466nMAssay Description:Binding affinity to human LYPLA1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetEpithelial cell adhesion molecule(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.472nMAssay Description:Binding affinity to human EPCAM incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Target26S proteasome non-ATPase regulatory subunit 5(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.486nMAssay Description:Binding affinity to human PSMD5 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.491nMAssay Description:Binding affinity to human EEF1G incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetNicotinate phosphoribosyltransferase(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.495nMAssay Description:Binding affinity to human NAPRT incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetLarge subunit GTPase 1 homolog(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.521nMAssay Description:Binding affinity to human LSG1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetSplicing factor U2AF 35 kDa subunit(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.531nMAssay Description:Binding affinity to human U2AF1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.546nMAssay Description:Binding affinity to human HSP90AB1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetCytochrome c1, heme protein, mitochondrial(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.550nMAssay Description:Binding affinity to human CYC1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.577nMAssay Description:Binding affinity to human COL14A1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.598nMAssay Description:Binding affinity to human UBQLN1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.606nMAssay Description:Binding affinity to human CDK4 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetSmall ribosomal subunit protein uS12(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.624nMAssay Description:Binding affinity to human RPS23 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetADP-ribosylation factor-like protein 1(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.716nMAssay Description:Binding affinity to human ARL1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.753nMAssay Description:Binding affinity to human NEK1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetDual specificity testis-specific protein kinase 2(Human)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.772nMAssay Description:Binding affinity to human TESK2 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetNuclear cap-binding protein subunit 1(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.799nMAssay Description:Binding affinity to human NCBP1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
TargetDnaJ homolog subfamily B member 12(Homo sapiens)
Johann Wolfgang Goethe University
Curated by ChEMBL
Johann Wolfgang Goethe University
Curated by ChEMBL
Affinity DataKd: 0.810nMAssay Description:Binding affinity to human DNAJB12 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.820nMAssay Description:Binding affinity to human IPO11 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair
Affinity DataKd: 0.852nMAssay Description:Binding affinity to human SDAD1 incubated for 45 mins by Kinobead based pull down assayMore data for this Ligand-Target Pair



3D Structure (crystal)