Compile Data Set for Download or QSAR
maximum 50k data
Found 21 Enz. Inhib. hit(s) with all data for entry = 50008318
LigandPNGBDBM247150((S,E)-2-Methyl-N-(2,2,2-trifluoro-1-(4-((5,5,5-tri...)
Affinity DataIC50:  0.200nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518061(CHEMBL4564881)
Affinity DataIC50:  0.300nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518066(CHEMBL4572662)
Affinity DataIC50:  0.380nMAssay Description:Inhibition of recombinant human MGAT2 using 2-monooleoyl glycerol/[1-14C]-oleoyl CoA as substrate after 30 mins by liquid scintillation counting meth...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518064(CHEMBL4463750)
Affinity DataIC50:  0.640nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM403538(US10335401, No. I-47)
Affinity DataIC50:  0.730nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM235244(US9365558, 67 | US9822074, 67)
Affinity DataIC50:  1nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518065(CHEMBL4577504)
Affinity DataIC50: <1nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518063(CHEMBL4465236)
Affinity DataIC50:  1.10nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM272063(US10065945, Example 57)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518069(CHEMBL4542050 | US11479538, Example 22)
Affinity DataIC50:  2nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518060(CHEMBL4455357)
Affinity DataIC50:  2.40nMAssay Description:Inhibition of recombinant mouse MGAT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50518071(CHEMBL3545611)
Affinity DataIC50:  3.80nMAssay Description:Inhibition of recombinant human MGAT2 expressed in sf9 cells using 2-monooleoyl glycerol/[14C]-oleoyl CoA as substrate by microscintillation counting...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518070(CHEMBL4466376)
Affinity DataIC50:  4nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50433269(CHEMBL2376303)
Affinity DataIC50:  6.30nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50518062(CHEMBL4441959)
Affinity DataIC50:  7nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518060(CHEMBL4455357)
Affinity DataIC50:  7.80nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50518059(CHEMBL4452833)
Affinity DataIC50:  19nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50518067(CHEMBL4560833)
Affinity DataIC50:  56nMAssay Description:Inhibition of recombinant human MGAT2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50518068(CHEMBL4535947)
Affinity DataIC50:  58nMAssay Description:Inhibition of recombinant human MGAT2 expressed in sf9 cells using 2-monooleoyl glycerol/[14C]-oleoyl CoA as substrate by microscintillation counting...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM152807(BDBM152808 | US8993568, 2)
Affinity DataIC50:  274nMAssay Description:Inhibition of recombinant human MGAT2 expressed in sf9 cells using 2-monooleoyl glycerol/[14C]-oleoyl CoA as substrate by microscintillation counting...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDiacylglycerol O-acyltransferase 2(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50518059(CHEMBL4452833)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibition of recombinant human DGAT2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed