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Found 6 Enz. Inhib. hit(s) with all data for entry = 50001754
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50366305(CHEBI:70328 | CHEMBL445599)
Affinity DataIC50:  500nMAssay Description:Inhibition of human p300 expressed in Escherichia coli incubated for 15 mins followed by [3H]acetyl-CoA/histone additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50366333(CHEMBL4166991)
Affinity DataIC50:  3.30E+3nMAssay Description:Inhibition of human p300 expressed in Escherichia coli incubated for 15 mins followed by [3H]acetyl-CoA/histone additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50366297(CHEMBL4173838)
Affinity DataIC50:  8.80E+3nMAssay Description:Inhibition of human p300 expressed in Escherichia coli incubated for 15 mins followed by [3H]acetyl-CoA/histone additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50366332(CHEMBL4162478)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human p300 expressed in Escherichia coli incubated for 15 mins followed by [3H]acetyl-CoA/histone additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50366313(CHEMBL4170395)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human p300 expressed in Escherichia coli incubated for 15 mins followed by [3H]acetyl-CoA/histone additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone acetyltransferase p300(Homo sapiens (Human))
Second Military Medical University

Curated by ChEMBL
LigandPNGBDBM50366309(CHEMBL4165919)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of human p300 expressed in Escherichia coli incubated for 15 mins followed by [3H]acetyl-CoA/histone additionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed