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Report error Found 30 Enz. Inhib. hit(s) with all data for entry = 50003266 Sort by
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50431886(CHEMBL1413473)
Affinity DataIC50: 4.90nMAssay Description:Inhibition of human recombinant BChE using butyrylthiocholine as substrate preincubated for 300 secs followed by substrate addition and measured for ...More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468744(CHEMBL4280947)
Affinity DataIC50: 9.5nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468733(CHEMBL4294570)
Affinity DataIC50: 11nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468736(CHEMBL4283585)
Affinity DataIC50: 14nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468741(CHEMBL4291165)
Affinity DataIC50: 19nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 22nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 23nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468739(CHEMBL4288890)
Affinity DataIC50: 28nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM11682(2,3-dihydroxybutanedioic acid; 3-[(1S)-1-(dimethyl...)
Affinity DataIC50: 30nMAssay Description:Inhibition of BChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468731(CHEMBL4287944)
Affinity DataIC50: 48nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468735(CHEMBL4288849)
Affinity DataIC50: 71nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468748(CHEMBL4277303)
Affinity DataIC50: 103nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8961(CHEMBL95 | Cognex | cid_1935 | CHEMBL1337960 | 1,2...)
Affinity DataIC50: 115nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min by...More data for this Ligand-Target Pair
In DepthDetails Article
PubMedPDB3D3D Structure (crystal)
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468743(CHEMBL4284357)
Affinity DataIC50: 135nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468742(CHEMBL4287764)
Affinity DataIC50: 229nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468732(CHEMBL4279606)
Affinity DataIC50: 237nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468737(CHEMBL4278201)
Affinity DataIC50: 266nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 300nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468747(CHEMBL4287511)
Affinity DataIC50: 460nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468734(CHEMBL4277107)
Affinity DataIC50: 635nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468740(CHEMBL4283974)
Affinity DataIC50: 1.61E+3nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468746(CHEMBL4294752)
Affinity DataIC50: 1.79E+3nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468745(CHEMBL4284141)
Affinity DataIC50: 2.49E+3nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetAcetylcholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM11682(2,3-dihydroxybutanedioic acid; 3-[(1S)-1-(dimethyl...)
Affinity DataIC50: 3.03E+3nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM8960(2-[(1-benzylpiperidin-4-yl)methyl]-5,6-dimethoxy-2...)
Affinity DataIC50: 4.15E+3nMAssay Description:Inhibition of BChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468730(CHEMBL4280532)
Affinity DataIC50: 6.92E+3nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM10404(galantamine | (1S,12S,14R)-9-methoxy-4-methyl-11-o...)
Affinity DataIC50: 7.00E+3nMAssay Description:Inhibition of BChE (unknown origin)More data for this Ligand-Target Pair
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468738(CHEMBL4292256)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured for 1 min b...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468733(CHEMBL4294570)
Affinity DataKi:  1.10nMAssay Description:Competitive inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetCholinesterase(Human)
University of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50468736(CHEMBL4283585)
Affinity DataKi:  1.70nMAssay Description:Competitive inhibition of human BChE using butyrylthiocholine iodide as substrate preincubated for 5 mins followed by substrate addition and measured...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed