Compile Data Set for Download or QSAR
Report error Found 121 Enz. Inhib. hit(s) with all data for entry = 50002465 Sort by
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458905(CHEMBL4208076)
Affinity DataEC50:  146nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458886(CHEMBL4217406)
Affinity DataEC50:  1.25E+3nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458884(CHEMBL4206798)
Affinity DataEC50:  71nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458906(CHEMBL4202758)
Affinity DataEC50:  18nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458907(CHEMBL4204245)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458899(CHEMBL4214230)
Affinity DataEC50:  5.76E+3nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458890(CHEMBL4218435)
Affinity DataEC50:  941nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458908(CHEMBL4216877)
Affinity DataEC50:  276nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458886(CHEMBL4217406)
Affinity DataEC50:  242nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458880(CHEMBL4209027)
Affinity DataEC50:  2.90E+3nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458882(CHEMBL4213948)
Affinity DataEC50:  1.73E+3nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458884(CHEMBL4206798)
Affinity DataEC50:  780nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458896(CHEMBL4211163)
Affinity DataEC50:  2.78E+3nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458904(CHEMBL4203290)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458889(CHEMBL4214942)
Affinity DataEC50:  139nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458898(CHEMBL4210525)
Affinity DataEC50:  194nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458897(CHEMBL4206281)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458901(CHEMBL4210242)
Affinity DataEC50:  4.93E+3nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458887(CHEMBL4212982)
Affinity DataEC50:  658nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458903(CHEMBL4218543)
Affinity DataEC50:  222nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458895(CHEMBL4202433)
Affinity DataEC50:  355nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458881(CHEMBL4215467)
Affinity DataEC50:  749nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458901(CHEMBL4210242)
Affinity DataEC50:  43nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458905(CHEMBL4208076)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458893(CHEMBL4212447)
Affinity DataEC50:  273nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458909(CHEMBL4207109)
Affinity DataEC50:  93nMAssay Description:Agonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458893(CHEMBL4212447)
Affinity DataEC50:  63nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458888(CHEMBL4205342)
Affinity DataEC50:  2nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458897(CHEMBL4206281)
Affinity DataEC50:  4nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458892(CHEMBL4208593)
Affinity DataEC50:  3nMAssay Description:Agonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458884(CHEMBL4206798)
Affinity DataIC50: 2nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458905(CHEMBL4208076)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458907(CHEMBL4204245)
Affinity DataIC50: 3nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458908(CHEMBL4216877)
Affinity DataIC50: 5nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458897(CHEMBL4206281)
Affinity DataIC50: 7nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458886(CHEMBL4217406)
Affinity DataIC50: 10nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458909(CHEMBL4207109)
Affinity DataIC50: 13nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458898(CHEMBL4210525)
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458906(CHEMBL4202758)
Affinity DataIC50: 27nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458882(CHEMBL4213948)
Affinity DataIC50: 42nMAssay Description:Antagonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458892(CHEMBL4208593)
Affinity DataIC50: 48nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458903(CHEMBL4218543)
Affinity DataIC50: 49nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458895(CHEMBL4202433)
Affinity DataIC50: 54nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458891(CHEMBL4203715)
Affinity DataIC50: 61nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458900(CHEMBL4205171)
Affinity DataIC50: 62nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor beta(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458884(CHEMBL4206798)
Affinity DataIC50: 69nMAssay Description:Antagonist activity at human ERbeta expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458882(CHEMBL4213948)
Affinity DataIC50: 72nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458904(CHEMBL4203290)
Affinity DataIC50: 149nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458893(CHEMBL4212447)
Affinity DataIC50: 166nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
TargetEstrogen receptor(Human)
Wuhan University

Curated by ChEMBL
LigandPNGBDBM50458887(CHEMBL4212982)
Affinity DataIC50: 428nMAssay Description:Antagonist activity at human ERalpha expressed in HEK293T cells after 24 hrs by ERE-based dual luciferase reporter gene assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails Article
PubMed
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