Compile Data Set for Download or QSAR
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Report error Found 9 Enz. Inhib. hit(s) with all data for entry = 50003272
TargetSerine/threonine-protein kinase B-raf(Mouse)
Nahda University

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  40nMAssay Description:Inhibition of mouse full length GST-tagged BRAF V600E mutant using recombinant human His6-tagged MEK1 as substrate preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Nahda University

Curated by ChEMBL
LigandPNGBDBM5446(CHEMBL553 | ERLOTINIB HYDROCHLORIDE | Erlotinib | ...)
Affinity DataIC50:  70nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank
MMDB
PDB3D3D Structure (crystal)

TargetEpidermal growth factor receptor(Human)
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468896(CHEMBL4279008)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468892(CHEMBL4289274)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468891(CHEMBL4286943)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetSerine/threonine-protein kinase B-raf(Mouse)
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468896(CHEMBL4279008)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of mouse full length GST-tagged BRAF V600E mutant using recombinant human His6-tagged MEK1 as substrate preincubated for 1 hr followed by ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468895(CHEMBL4290355)
Affinity DataIC50:  5.60E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468894(CHEMBL4282482)
Affinity DataIC50:  7.20E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed

TargetEpidermal growth factor receptor(Human)
Nahda University

Curated by ChEMBL
LigandPNGBDBM50468893(CHEMBL4286998)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of His6-tagged recombinant EGFR cytoplasmic domain (645 to 1186 residues) (unknown origin) expressed in baculovirus infected Sf9 insect ce...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed