Compile Data Set for Download or QSAR
Report error Found 52 Enz. Inhib. hit(s) with all data for entry = 50002820
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463446BDBM50463446(CHEMBL4244422)
Affinity DataEC50:  230nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463446BDBM50463446(CHEMBL4244422)
Affinity DataIC50: 260nMAssay Description:Antagonist activity at rat TRPA1 expressed in HEK293 cells assessed as inhibition of AITC-induced increase in intracellular calcium level pretreated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataIC50: 270nMAssay Description:Antagonist activity at rat TRPA1 expressed in HEK293 cells assessed as inhibition of AITC-induced increase in intracellular calcium level pretreated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataEC50:  290nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463443BDBM50463443(CHEMBL4241477)
Affinity DataIC50: 320nMAssay Description:Antagonist activity at rat TRPA1 expressed in HEK293 cells assessed as inhibition of AITC-induced increase in intracellular calcium level pretreated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463443BDBM50463443(CHEMBL4241477)
Affinity DataEC50:  350nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataIC50: 450nMAssay Description:Antagonist activity at rat TRPA1 expressed in HEK293 cells assessed as inhibition of AITC-induced increase in intracellular calcium level pretreated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataEC50:  490nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463442BDBM50463442(CHEMBL4242719)
Affinity DataEC50:  1.30E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463442BDBM50463442(CHEMBL4242719)
Affinity DataIC50: 1.70E+3nMAssay Description:Antagonist activity at rat TRPA1 expressed in HEK293 cells assessed as inhibition of AITC-induced increase in intracellular calcium level pretreated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataEC50:  1.80E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463444BDBM50463444(CHEMBL4238978)
Affinity DataEC50:  2.00E+3nMAssay Description:Agonist activity at rat TRPA1 expressed in HEK293 cells assessed as increase in intracellular calcium level by fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463444BDBM50463444(CHEMBL4238978)
Affinity DataIC50: 2.30E+3nMAssay Description:Antagonist activity at rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced increase in intracellular calcium level pretreated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataEC50:  2.60E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataEC50:  3.30E+3nMAssay Description:Agonist activity at rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataIC50: 3.90E+3nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataIC50: 4.30E+3nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463443BDBM50463443(CHEMBL4241477)
Affinity DataIC50: 4.50E+3nMAssay Description:Antagonist activity at rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced increase in intracellular calcium level pretreated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataEC50:  4.70E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily A member 1(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463444BDBM50463444(CHEMBL4238978)
Affinity DataIC50: 4.80E+3nMAssay Description:Antagonist activity at rat TRPA1 expressed in HEK293 cells assessed as inhibition of AITC-induced increase in intracellular calcium level pretreated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463442BDBM50463442(CHEMBL4242719)
Affinity DataEC50:  4.90E+3nMAssay Description:Agonist activity at human TRPV1 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence ass...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataEC50:  5.80E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataIC50: 5.90E+3nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463442BDBM50463442(CHEMBL4242719)
Affinity DataEC50:  6.40E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataEC50:  6.70E+3nMAssay Description:Agonist activity at rat TRPV3 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataIC50: 7.10E+3nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463444BDBM50463444(CHEMBL4238978)
Affinity DataIC50: 7.20E+3nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of icilin-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataIC50: 8.00E+3nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of thymol-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463446BDBM50463446(CHEMBL4244422)
Affinity DataEC50:  8.40E+3nMAssay Description:Agonist activity at rat TRPV2 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataIC50: 1.28E+4nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of thymol-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataIC50: 1.37E+4nMAssay Description:Antagonist activity at rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced increase in intracellular calcium level pretreated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataIC50: 1.71E+4nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of icilin-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463443BDBM50463443(CHEMBL4241477)
Affinity DataEC50:  1.80E+4nMAssay Description:Agonist activity at rat TRPV4 expressed in HEK293 cells assessed as increase in intracellular calcium level by Fluo-4-AM dye based fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463442BDBM50463442(CHEMBL4242719)
Affinity DataIC50: 3.70E+4nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463442BDBM50463442(CHEMBL4242719)
Affinity DataIC50: 3.97E+4nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463442BDBM50463442(CHEMBL4242719)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of thymol-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463446BDBM50463446(CHEMBL4244422)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of thymol-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463443BDBM50463443(CHEMBL4241477)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of thymol-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463442BDBM50463442(CHEMBL4242719)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of icilin-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463443BDBM50463443(CHEMBL4241477)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463442BDBM50463442(CHEMBL4242719)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced increase in intracellular calcium level pretreated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel, subfamily V, member 3(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463444BDBM50463444(CHEMBL4238978)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of thymol-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463445BDBM50463445(CHEMBL4238545)
Affinity DataIC50: 5.00E+4nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of icilin-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 2(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463447BDBM50463447(CHEMBL4249046)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat TRPV2 expressed in HEK293 cells assessed as inhibition of LPC-induced increase in intracellular calcium level pretreated f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily M member 8(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463443BDBM50463443(CHEMBL4241477)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat TRPM8 expressed in HEK293 cells assessed as inhibition of icilin-induced increase in intracellular calcium level pretreate...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463443BDBM50463443(CHEMBL4241477)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463444BDBM50463444(CHEMBL4238978)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463444BDBM50463444(CHEMBL4238978)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 1(Human)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463446BDBM50463446(CHEMBL4244422)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at human TRPV1 expressed in HEK293 cells assessed as inhibition of capsaicin-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
TargetTransient receptor potential cation channel subfamily V member 4(Rat)
University of Naples Federico II

Curated by ChEMBL
LigandChemical structure of BindingDB Monomer ID 50463446BDBM50463446(CHEMBL4244422)
Affinity DataIC50: 1.00E+5nMAssay Description:Antagonist activity at rat TRPV3 expressed in HEK293 cells assessed as inhibition of GSK1016790A-induced increase in intracellular calcium level pret...More data for this Ligand-Target Pair
In Depth
Date in BDB:
8/17/2020
Entry Details Article
PubMed
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