Report error Found 10 Enz. Inhib. hit(s) with all data for entry = 50009522
Affinity DataKi: 150nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 150nMAssay Description:Displacement of [3H]CP55940 from human CB2 expressed in CHOK1 cell membranes after 2 hrs by liquid scintillation counting methodMore data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at human alpha7 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced currents at -70 mV hold...More data for this Ligand-Target Pair
TargetNeuronal acetylcholine receptor subunit alpha-7(Human)
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Affinity DataIC50: 3.10E+3nMAssay Description:Antagonist activity at human alpha7 nACHR expressed in Xenopus laevis oocytes assessed as inhibition of acetylcholine-induced currents at -70 mV hold...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Antagonist activity at TRPA1 (unknown origin) expressed in Xenopus laevis oocytes assessed as inhibition of mustard oil-induced currents by two-elect...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Affinity DataIC50: 3.00E+5nMAssay Description:Antagonist activity at TRPA1 (unknown origin) expressed in Xenopus laevis oocytes assessed as inhibition of mustard oil-induced currents by two-elect...More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Agonist activity at recombinant human Cb2 receptor expressed in CHOK1 cells assessed as inhibition of forskolin-stimulated cAMP levels measured up to...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Affinity DataEC50: 3.30E+4nMAssay Description:Agonist activity at human TRPA1More data for this Ligand-Target Pair
Affinity DataEC50: 1.90E+3nMAssay Description:Agonist activity at recombinant human Cb2 receptor expressed in CHOK1 cells assessed as inhibition of forskolin-stimulated cAMP levels measured up to...More data for this Ligand-Target Pair
TargetTransient receptor potential cation channel subfamily A member 1(Human)
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Univerisity of Eastern Finland (Uef)
Curated by ChEMBL
Affinity DataEC50: 3.30E+4nMAssay Description:Agonist activity at human TRPA1More data for this Ligand-Target Pair
